SCHEMBL383668

SCHEMBL383668

COc1cc(C(=O)NC[C@@](NS(=O)(=O)c2ccc(C(=O)O)cc2)(C(=O)O)C(C)(C)C)ccc1N1CCC(Nc2ncccn2)CC1

nearest known ligand 0.48

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 7/20 0.48
ITGAV P06756 7/20 0.48
ITGA2B P08514 7/20 0.48
DRD2 P14416 1/20 0.38
DRD3 P35462 1/20 0.38
ALDH1A1 P00352 4/20 0.38
LMNA P02545 2/20 0.38
HTT P42858 2/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
USP30 Q70CQ3 1/20 0.36
TDP1 Q9NUW8 1/20 0.35
USP2 O75604 1/20 0.35
TSHR P16473 1/20 0.35
PTK2 Q05397 1/20 0.34
ROCK2 O75116 1/20 0.34
KDM4E B2RXH2 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL382191 0.96 ITGB3 (0.53) ITGB3ITGAVITGA2BDRD2DRD3
SCHEMBL383098 0.86 ITGB3 (0.50) ITGB3ITGAVITGA2B
SCHEMBL382826 0.85 ITGB3 (0.51) ITGB3ITGAVITGA2BALDH1A1LMNA
SCHEMBL383666 0.85 ITGB3 (0.46) ITGB3ITGAVITGA2BDRD2DRD3
SCHEMBL7650917 0.85 ITGB3 (0.47) ITGB3ITGAVITGA2BDRD2DRD3
SCHEMBL6497874 0.84 ITGB3 (0.44) ITGB3ITGAVITGA2BLMNA
SCHEMBL6497211 0.84 DRD2 (0.41) ITGB3ITGAVITGA2BDRD2DRD3
SCHEMBL383161 0.82 ITGB3 (0.47) ITGB3ITGAVITGA2BDRD2DRD3
SCHEMBL382694 0.82 ITGB3 (0.46) ITGB3ITGAVITGA2BDRD2DRD3
SCHEMBL382492 0.82 ITGB3 (0.70) ITGB3ITGAVITGA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1074543-B1 AMINOPIPERIDINE DERIVATIVES AS INTEGRIN ALPHA V BETA 3 ANTAGONISTS MEIJI SEIKA PHARMA CO LTD (JP) 2012-01-25 EP disclosed