SCHEMBL3836802

SCHEMBL3836802

CCCc1cccc(C#Cc2ccccc2)c1

nearest known ligand 0.56

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PTGES O14684 6/20 0.50
FFAR1 O14842 4/20 0.46
CYP2D6 P10635 1/20 0.46
HRH3 Q9Y5N1 1/20 0.46
APP P05067 1/20 0.46
DRD2 P14416 1/20 0.42
OPRM1 P35372 1/20 0.42
DRD3 P35462 1/20 0.42
OPRD1 P41143 1/20 0.42
OPRK1 P41145 1/20 0.42
ASIC3 Q9UHC3 1/20 0.42
KIF11 P52732 1/20 0.42
KAT6A Q92794 1/20 0.41
KCNH2 Q12809 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3837565 0.90 PTGES (0.46) PTGESFFAR1CYP2D6HRH3DRD2
SCHEMBL3859050 0.87 CA12 (0.47) PTGESFFAR1KCNH2
SCHEMBL3841194 0.87 FFAR1 (0.44) PTGESFFAR1CYP2D6HRH3DRD2
SCHEMBL3859573 0.86 PTGES (0.44) PTGESFFAR1CYP2D6HRH3
SCHEMBL3864253 0.84 ASIC3 (0.47) PTGESFFAR1ASIC3
SCHEMBL3843357 0.84 GRM5 (0.48) PTGESFFAR1CYP2D6HRH3DRD2
SCHEMBL27874223 0.84 TP53 (0.52) PTGESFFAR1CYP2D6HRH3APP
SCHEMBL3839454 0.83 FFAR1 (0.47) PTGESFFAR1CYP2D6HRH3
SCHEMBL3859036 0.82 FFAR1 (0.47) PTGESFFAR1CYP2D6HRH3DRD2
SCHEMBL2833040 0.82 FFAR1 (0.58) FFAR1APPASIC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2111223-A1 AMINE DERIVATIVE COMPOUNDS FOR TREATING OPHTHALMIC DISEASES AND DISORDERS Acucela, Inc. (US) 2009-10-28 EP disclosed
WO-2009058216-A1 AMINE DERIVATIVE COMPOUNDS FOR TREATING OPHTHALMIC DISEASES AND DISORDERS ACUCELA, INC. (US) 2009-05-07 WO disclosed