SCHEMBL3864253

SCHEMBL3864253

CCCc1cccc(C#Cc2ccc3ccccc3c2)c1

nearest known ligand 0.47

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ASIC3 Q9UHC3 2/20 0.47
ACACB O00763 1/20 0.43
CYP1A2 P05177 2/20 0.42
CYP2A6 P11509 1/20 0.42
BCHE P06276 2/20 0.40
PTGES O14684 1/20 0.39
CYP1A1 P04798 1/20 0.39
CYP1B1 Q16678 1/20 0.39
FFAR1 O14842 2/20 0.38
SIGMAR1 Q99720 1/20 0.38
CTSS P25774 1/20 0.37
CTSK P43235 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3836802 0.84 PTGES (0.50) ASIC3PTGESFFAR1
SCHEMBL2754684 0.81 ASIC3 (0.45) ASIC3ACACBCYP1A2FFAR1SIGMAR1
SCHEMBL236242 0.81 ASIC3 (0.53) ASIC3ACACBCYP1A2SIGMAR1
SCHEMBL3859050 0.80 CA12 (0.47) PTGESFFAR1
SCHEMBL9742625 0.80 ASIC3 (0.53) ASIC3ACACBCYP1A2CYP2A6FFAR1
SCHEMBL3837565 0.79 PTGES (0.46) ASIC3PTGESFFAR1CTSSCTSK
SCHEMBL9742914 0.77 ASIC3 (0.50) ASIC3ACACBCYP1A2CYP2A6
SCHEMBL3841194 0.77 FFAR1 (0.44) CYP1A2PTGESFFAR1SIGMAR1
SCHEMBL140016 0.77 CYP1A2 (0.68) CYP1A2CYP2A6BCHESIGMAR1
SCHEMBL5573799 0.76 ASIC3 (0.53) ASIC3ACACBCYP1A2CYP2A6CYP1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2076122-A2 ALKYNYL PHENYL DERIVATIVE COMPOUNDS FOR TREATING OPHTHALMIC DISEASES AND DISORDERS Acucela, Inc. (US) 2009-07-08 EP disclosed
WO-2009005794-A2 ALKYNYL PHENYL DERIVATIVE COMPOUNDS FOR TREATING OPHTHALMIC DISEASES AND DISORDERS ACUCELA, INC. (US) 2009-01-08 WO disclosed