SCHEMBL3837692

SCHEMBL3837692

COC(OC)c1ccc(C(=O)NC(C)(C)c2ccccc2)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 2/20 0.49
ROCK1 Q13464 1/20 0.49
IMPDH2 P12268 1/20 0.46
ADAMTS4 O75173 1/20 0.45
ADAMTS5 Q9UNA0 1/20 0.45
PHGDH O43175 1/20 0.42
POLB P06746 1/20 0.41
KMT2A Q03164 2/20 0.41
MEN1 O00255 1/20 0.41
ALPL P05186 1/20 0.40
GLA P06280 1/20 0.40
ALPI P09923 1/20 0.40
ALPG P10696 1/20 0.40
EGLN1 Q9GZT9 1/20 0.40
TACR3 P29371 1/20 0.40
NR1H4 Q96RI1 1/20 0.40
HDAC1 Q13547 2/20 0.40
HDAC8 Q9BY41 2/20 0.40
HDAC6 Q9UBN7 2/20 0.40
ALDH1A1 P00352 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL94229 0.82 IMPDH2 (0.52) ROCK2ROCK1IMPDH2ADAMTS4ADAMTS5
SCHEMBL3039120 0.81 POLB (0.58) ROCK2ROCK1IMPDH2ADAMTS4ADAMTS5
SCHEMBL3834428 0.81 ROCK2 (0.49) ROCK2ROCK1IMPDH2ADAMTS4ADAMTS5
SCHEMBL3836272 0.80 RAB9A (0.57) ROCK2IMPDH2ADAMTS4ADAMTS5POLB
SCHEMBL3838597 0.79 IMPDH2 (0.52) ROCK2ROCK1IMPDH2ADAMTS4ADAMTS5
SCHEMBL3836954 0.77 IMPDH2 (0.51) ROCK2ROCK1IMPDH2ADAMTS4ADAMTS5
SCHEMBL3835811 0.77 POLB (0.56) ROCK2IMPDH2ADAMTS4ADAMTS5PHGDH
SCHEMBL3835902 0.77 PPARG (0.52) ROCK2IMPDH2ADAMTS4ADAMTS5PHGDH
SCHEMBL27476988 0.77 NPC1 (0.50) POLBHDAC8HDAC6ALDH1A1
SCHEMBL3840595 0.75 KDM4E (0.49) ROCK2ROCK1IMPDH2ADAMTS4ADAMTS5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2108642-A1 JAK INHIBITOR Kyowa Hakko Kirin Co., Ltd. (JP) 2009-10-14 EP disclosed