SCHEMBL3841735

SCHEMBL3841735

O=C(O)Cc1cc(-c2cccs2)c[nH]c1=O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 1/20 0.46
ALDH1A1 P00352 2/20 0.41
PPARG P37231 2/20 0.41
KDM4E B2RXH2 1/20 0.41
NCOA2 Q15596 1/20 0.41
NCOA1 Q15788 1/20 0.41
RXFP1 Q9HBX9 1/20 0.41
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
GPR17 Q13304 1/20 0.39
GRK6 P43250 1/20 0.38
HTR1D P28221 1/20 0.38
HTR1B P28222 1/20 0.38
ACMSD Q8TDX5 2/20 0.38
FFAR1 O14842 2/20 0.37
PPARA Q07869 1/20 0.37
ERCC1 P07992 1/20 0.36
FEN1 P39748 1/20 0.36
ERCC4 Q92889 1/20 0.36
NPC1 O15118 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3841574 0.81 ALDH1A1 (0.43) PTPN1ALDH1A1KDM4EKMT2AHTR1D
SCHEMBL3846364 0.72 IDO1 (0.46) ALDH1A1KDM4EMEN1KMT2ANPC1
SCHEMBL5183298 0.69 KDM4E (0.52) ALDH1A1KDM4ERXFP1FEN1
SCHEMBL6516216 0.69 LTA4H (0.59) ALDH1A1PPARGKDM4ENCOA2NCOA1
SCHEMBL6393707 0.69 FFAR1 (0.57) ALDH1A1PPARGKDM4ENCOA2NCOA1
SCHEMBL4048685 0.68 LTA4H (0.54) PTPN1ALDH1A1PPARGKDM4ENCOA2
SCHEMBL5053028 0.68 ALDH1A1 (0.47) PTPN1ALDH1A1PPARGKDM4ENCOA2
SCHEMBL352568 0.68 ALDH1A1 (0.47) PTPN1ALDH1A1PPARGKDM4ENCOA2
SCHEMBL3844258 0.67 ERCC1 (0.50) ALDH1A1KDM4EMEN1KMT2AERCC1
SCHEMBL9450326 0.66 ALDH1A1 (0.44) ALDH1A1PPARGKDM4ENCOA2NCOA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2114898-A2 NITROGEN-CONTAINING HETEROCYCLYL KETONES AND THEIR USE AS C-MET INHIBITORS Amgen Inc. (US) 2009-11-11 EP disclosed
WO-2008103277-A2 NITROGEN-CONTAINING HETEROCYCLYL KETONES AND THEIR USE AS C-MET INHIBITORS AMGEN INC. (US) 2008-08-28 WO disclosed