SCHEMBL3842349

SCHEMBL3842349

CCC(O)C(C)Cc1cccc(C(O)CCN)c1

nearest known ligand 0.54

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 1/20 0.54
ADRB2 P07550 4/20 0.36
NOS1 P29475 1/20 0.36
NOS2 P35228 1/20 0.36
LMNA P02545 1/20 0.34
PNMT P11086 2/20 0.33
PGK1 P00558 1/20 0.33
PGK2 P07205 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10287473 0.84 NOS1 (0.39) ADRB2NOS1NOS2PNMTPGK1
SCHEMBL17277380 0.81 CYP3A4 (0.41) NOS1NOS2LMNAPNMTPGK1
SCHEMBL612758 0.77 NOS1 (0.40) NOS1NOS2PNMTPGK1PGK2
SCHEMBL611386 0.76 NOS1 (0.33) ADRB2NOS1NOS2PNMT
SCHEMBL13959620 0.76 PRSS1 (0.41) ADRB2NOS1NOS2PNMTPGK1
SCHEMBL14642896 0.75 LPL (0.42) NOS1NOS2
SCHEMBL3839058 0.75 NOS1 (0.38) NOS1NOS2PNMT
SCHEMBL610891 0.74 GRIN2D (0.40) NOS1NOS2LMNAPNMT
SCHEMBL27836303 0.74 PNMT (0.39) ADRB2NOS1NOS2LMNAPNMT
SCHEMBL28043377 0.74 PGK1 (0.42) NOS1NOS2PNMTPGK1PGK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2111223-A1 AMINE DERIVATIVE COMPOUNDS FOR TREATING OPHTHALMIC DISEASES AND DISORDERS Acucela, Inc. (US) 2009-10-28 EP disclosed
WO-2009058216-A1 AMINE DERIVATIVE COMPOUNDS FOR TREATING OPHTHALMIC DISEASES AND DISORDERS ACUCELA, INC. (US) 2009-05-07 WO disclosed