SCHEMBL3844597

SCHEMBL3844597

Cc1ccc(CNc2ccccc2)cn1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LTA4H P09960 1/20 0.59
GAA P10253 2/20 0.50
HTT P42858 1/20 0.50
ALDH1A1 P00352 1/20 0.50
MEN1 O00255 1/20 0.50
CYP1A2 P05177 1/20 0.50
CYP3A4 P08684 1/20 0.50
CYP2C9 P11712 1/20 0.50
CYP2C19 P33261 1/20 0.50
KMT2A Q03164 1/20 0.50
RAB9A P51151 1/20 0.50
NAMPT P43490 1/20 0.48
HDAC1 Q13547 1/20 0.48
AURKA O14965 1/20 0.46
ABL1 P00519 1/20 0.46
NTRK1 P04629 1/20 0.46
LCK P06239 1/20 0.46
CSF1R P07333 1/20 0.46
RET P07949 1/20 0.46
MET P08581 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4592530 0.84 GAA (0.54) GAAHTTALDH1A1MEN1KMT2A
SCHEMBL4740818 0.83 AURKA (0.65) GAAHTTALDH1A1MEN1CYP1A2
SCHEMBL2500333 0.83 GAA (0.68) LTA4HGAAHTTALDH1A1MEN1
SCHEMBL16601601 0.82 HTT (0.59) LTA4HHTTALDH1A1RAB9AHDAC1
SCHEMBL13090580 0.79 KDM4E (0.72) LTA4HGAAALDH1A1MEN1CYP1A2
SCHEMBL30862011 0.79 KDM4E (0.72) LTA4HGAAALDH1A1MEN1CYP1A2
SCHEMBL2065031 0.76 CYP1A2 (0.69) LTA4HHTTALDH1A1MEN1CYP1A2
SCHEMBL4739798 0.76 LTA4H (0.47) LTA4HGAAHTTALDH1A1MEN1
SCHEMBL3038971 0.75 GAA (0.45) GAAMEN1CYP3A4KMT2ANAMPT
SCHEMBL1624682 0.75 HTT (0.84) GAAHTTALDH1A1MEN1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2099800-A1 7-SUBSTITUTED PURINE DERIVATIVES FOR IMMUNOSUPPRESSION Pharmacopeia, LLC (US) 2009-09-16 EP disclosed
WO-2008060301-A1 7-SUBSTITUTED PURINE DERIVATIVES FOR IMMUNOSUPPRESSION PHARMACOPEIA , LLC (US) 2008-05-22 WO disclosed