SCHEMBL3848964

SCHEMBL3848964

CCOC(=O)c1cc(-c2ncnc3ccc(-c4cnn(C(c5ccccc5)(c5ccccc5)c5ccccc5)c4)cc23)ccc1F

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CAMKK1 Q8N5S9 3/20 0.39
CAMKK2 Q96RR4 3/20 0.39
JAK3 P52333 9/20 0.38
JAK2 O60674 7/20 0.38
KDM4E B2RXH2 2/20 0.38
HPGD P15428 2/20 0.38
HSD17B10 Q99714 2/20 0.38
TSHR P16473 1/20 0.38
CASP1 P29466 1/20 0.38
CASP7 P55210 1/20 0.38
IRAK4 Q9NWZ3 1/20 0.38
RXFP1 Q9HBX9 1/20 0.37
MAPT P10636 2/20 0.36
NPC1 O15118 2/20 0.35
ALDH1A1 P00352 1/20 0.35
RAB9A P51151 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
PKM P14618 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3846919 0.94 NPC1 (0.43) CAMKK1CAMKK2JAK3JAK2KDM4E
SCHEMBL3848535 0.88 CAMKK1 (0.45) CAMKK1CAMKK2
SCHEMBL3847105 0.83 CAMKK2 (0.47) CAMKK1CAMKK2
SCHEMBL3847597 0.80 MAPT (0.40) CAMKK1CAMKK2KDM4ETSHRRXFP1
SCHEMBL3846835 0.79 MAPT (0.41) KDM4EHPGDHSD17B10MAPTALDH1A1
SCHEMBL3847931 0.77 AURKB (0.43) CAMKK1CAMKK2KDM4EHPGDHSD17B10
SCHEMBL3846925 0.77 JAK3 (0.48) CAMKK1CAMKK2JAK3JAK2KDM4E
SCHEMBL3845583 0.75 PKM (0.43) KDM4EHPGDHSD17B10TSHRCASP1
SCHEMBL3845338 0.74 LMNA (0.40) CAMKK1CAMKK2KDM4EHPGDHSD17B10
SCHEMBL3846747 0.73 RPS6KB2 (0.39) CAMKK1CAMKK2KDM4ENPC1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2048142-A2 Nitrogen-containing condensed cyclic compound having a pyrazolyl group as a substituent group and pharmaceutical composition thereof Eisai R&D Management Co., Ltd. (JP) 2009-04-15 EP disclosed
EP-1382603-B1 NITROGENOUS FUSED-RING COMPOUND HAVING PYRAZOLYL GROUP AS SUBSTITUENT AND MEDICINAL COMPOSITION THEREOF EISAI R&D MAN CO LTD (JP) 2008-07-23 EP disclosed
US-7074801-B1 Nitrogen-containing condensed cyclic compound having a pyrazolyl group as a substituent group and pharmaceutical composition thereof EISAI CO., LTD. (JP) 2006-07-11 US disclosed
EP-1382603-A1 NITROGENOUS FUSED−RING COMPOUND HAVING PYRAZOLYL GROUP AS SUBSTITUENT AND MEDICINAL COMPOSITION THEREOF Eisai Co., Ltd. (JP) 2004-01-21 EP disclosed