SCHEMBL3851773

SCHEMBL3851773

Cc1cc(NC(=O)c2ccc(Br)cc2F)on1

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.70
SMN1; SMN2 Q16637 4/20 0.70
GLA P06280 1/20 0.70
NPC1 O15118 2/20 0.51
RAB9A P51151 2/20 0.51
LMNA P02545 1/20 0.51
GAA P10253 1/20 0.51
KMT2A Q03164 1/20 0.51
PKM P14618 1/20 0.48
ATF1 P18846 1/20 0.47
NFKB1 P19838 1/20 0.47
MAPT P10636 1/20 0.47
THRB P10828 1/20 0.47
DGAT1 O75907 1/20 0.44
MAPK7 Q13164 1/20 0.44
GPR27 Q9NS67 1/20 0.43
SORT1 Q99523 5/20 0.43
HDAC4 P56524 1/20 0.42
HDAC6 Q9UBN7 1/20 0.42
FLT1 P17948 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3849262 0.80 RAB9A (0.57) ALDH1A1SMN1; SMN2NPC1RAB9ALMNA
SCHEMBL18420793 0.73 SMN1; SMN2 (0.66) ALDH1A1SMN1; SMN2NPC1RAB9ALMNA
SCHEMBL29803616 0.72 NPC1 (0.65) ALDH1A1SMN1; SMN2NPC1RAB9ALMNA
SCHEMBL24670566 0.72 NPC1 (0.65) ALDH1A1SMN1; SMN2NPC1RAB9ALMNA
SCHEMBL31511667 0.72 NPC1 (0.59) ALDH1A1SMN1; SMN2NPC1RAB9ALMNA
SCHEMBL1648482 0.72 DGAT1 (0.59) ALDH1A1SMN1; SMN2NPC1RAB9ALMNA
SCHEMBL13485811 0.71 DGAT1 (0.63) ALDH1A1SMN1; SMN2NPC1RAB9ALMNA
SCHEMBL27007857 0.71 DGAT1 (0.63) ALDH1A1SMN1; SMN2NPC1RAB9ALMNA
SCHEMBL3345916 0.71 DGAT1 (0.54) ALDH1A1SMN1; SMN2NPC1RAB9ALMNA
SCHEMBL3845645 0.71 SORT1 (0.73) ALDH1A1SMN1; SMN2GLANPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2048142-A2 Nitrogen-containing condensed cyclic compound having a pyrazolyl group as a substituent group and pharmaceutical composition thereof Eisai R&D Management Co., Ltd. (JP) 2009-04-15 EP disclosed
EP-1382603-B1 NITROGENOUS FUSED-RING COMPOUND HAVING PYRAZOLYL GROUP AS SUBSTITUENT AND MEDICINAL COMPOSITION THEREOF EISAI R&D MAN CO LTD (JP) 2008-07-23 EP disclosed
US-7074801-B1 Nitrogen-containing condensed cyclic compound having a pyrazolyl group as a substituent group and pharmaceutical composition thereof EISAI CO., LTD. (JP) 2006-07-11 US disclosed
EP-1382603-A1 NITROGENOUS FUSED−RING COMPOUND HAVING PYRAZOLYL GROUP AS SUBSTITUENT AND MEDICINAL COMPOSITION THEREOF Eisai Co., Ltd. (JP) 2004-01-21 EP disclosed