SCHEMBL3852258

SCHEMBL3852258

CCc1nc(C(C)=O)no1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
APOBEC3A P31941 2/20 0.35
APOBEC3G Q9HC16 2/20 0.35
KDM4E B2RXH2 2/20 0.35
HSD17B10 Q99714 2/20 0.35
ALOX15 P16050 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
ACACB O00763 1/20 0.32
ACACA Q13085 1/20 0.32
ALDH1A1 P00352 2/20 0.31
MEN1 O00255 1/20 0.31
TP53 P04637 1/20 0.31
GAA P10253 1/20 0.31
MAPT P10636 1/20 0.31
HPGD P15428 1/20 0.31
RAB9A P51151 1/20 0.31
KMT2A Q03164 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
SMPD1 P17405 3/20 0.31
HCRTR1 O43613 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13429229 0.82 SMPD1 (0.32) SMPD1
SCHEMBL17660397 0.72 RAB9A (0.47) APOBEC3AAPOBEC3GKDM4EHSD17B10ALOX15
SCHEMBL7263917 0.72 HSD17B10 (0.42) APOBEC3AAPOBEC3GKDM4EHSD17B10ALOX15
SCHEMBL1828616 0.71
SCHEMBL23635941 0.71 KDM4E (0.39) APOBEC3AAPOBEC3GKDM4EHSD17B10ALOX15
SCHEMBL6124859 0.69
SCHEMBL12705 0.66
SCHEMBL18141918 0.64 APOBEC3A (0.54) APOBEC3AAPOBEC3GKDM4EHSD17B10ALOX15
SCHEMBL265221 0.64 KDM4E (0.36) APOBEC3AAPOBEC3GKDM4EHSD17B10ALOX15
Ammonia Solution, Strong SCHEMBL3447928 0.64

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7576220-B2 Method of producing 1,2,4-oxadiazole derivatives RIKKYO GAKUIN (JP) 2009-08-18 US claimed
US-20080086009-A1 Method of producing 1,2,4-oxadiazole derivatives RIKKYO GAKUIN (JP) 2008-04-10 US claimed
US-7576220-B2 Method of producing 1,2,4-oxadiazole derivatives RIKKYO GAKUIN (JP) 2009-08-18 US disclosed
US-20080086009-A1 Method of producing 1,2,4-oxadiazole derivatives RIKKYO GAKUIN (JP) 2008-04-10 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080086009-A1 Method of producing 1,2,4-oxadiazole derivatives NOS1, NOS2, NOS3 APOBEC3A 420/4885APOBEC3G 794/4885KDM4E 2292/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.