SCHEMBL3852729

SCHEMBL3852729

Cc1n[nH]cc1-c1ccc2nccc(N3CCN(C(=O)N4CCOCC4)CC3)c2c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.43
AKR1C3 P42330 8/20 0.43
IDE P14735 1/20 0.40
KDM4E B2RXH2 1/20 0.40
HPGD P15428 1/20 0.40
HSD17B10 Q99714 1/20 0.40
GAA P10253 1/20 0.40
MAPT P10636 1/20 0.40
LMNA P02545 1/20 0.39
BMPR1B O00238 1/20 0.39
PDGFRB P09619 1/20 0.39
KIT P10721 1/20 0.39
PDGFRA P16234 1/20 0.39
BMPR1A P36894 1/20 0.39
ACVR1B P36896 1/20 0.39
TGFBR1 P36897 1/20 0.39
ACVRL1 P37023 1/20 0.39
ACVR1 Q04771 1/20 0.39
PIK3CA P42336 2/20 0.39
CLK1 P49759 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL5852245 0.99 ALDH1A1 (0.43) ALDH1A1AKR1C3IDEKDM4EHPGD
SCHEMBL3853295 0.87 IDE (0.42) ALDH1A1IDEMAPTPDGFRBCLK1
SCHEMBL3847156 0.86 AKR1C3 (0.43) ALDH1A1AKR1C3KDM4EHPGDHSD17B10
SCHEMBL3852919 0.85 MEN1 (0.46) ALDH1A1IDEMAPTPDGFRBACVR1
Hydrochloric Acid SCHEMBL3853045 0.83 MTNR1B (0.46) IDEKDM4EMAPTPDGFRBKIT
SCHEMBL3851448 0.82 NCF1 (0.45) ALDH1A1KDM4EHPGDHSD17B10LMNA
SCHEMBL3852118 0.81 DPP4 (0.41) IDEPDGFRBPIK3CANCF1
Hydrochloric Acid SCHEMBL5852112 0.81 NCF1 (0.44) ALDH1A1KDM4EHPGDHSD17B10LMNA
Hydrochloric Acid SCHEMBL3856136 0.80 PDGFRB (0.56) KDM4EGAAMAPTPDGFRB
SCHEMBL3854528 0.80 DPP4 (0.40) IDEPIK3CACLK1NCF1PIK3CD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2048142-A2 Nitrogen-containing condensed cyclic compound having a pyrazolyl group as a substituent group and pharmaceutical composition thereof Eisai R&D Management Co., Ltd. (JP) 2009-04-15 EP disclosed
EP-1382603-B1 NITROGENOUS FUSED-RING COMPOUND HAVING PYRAZOLYL GROUP AS SUBSTITUENT AND MEDICINAL COMPOSITION THEREOF EISAI R&D MAN CO LTD (JP) 2008-07-23 EP disclosed