SCHEMBL38530

SCHEMBL38530

N#CNC(=O)c1cc2nc(Cc3cccc(Cl)c3)[nH]c(=O)c2s1

nearest known ligand 0.73

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE5A O76074 4/20 0.73
PDE9A O76083 1/20 0.43
PDE1A P54750 1/20 0.43
PDE1B Q01064 1/20 0.43
PDE1C Q14123 1/20 0.43
MAPT P10636 3/20 0.42
RAB9A P51151 3/20 0.41
KDM4E B2RXH2 2/20 0.41
LMNA P02545 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
CDC7 O00311 4/20 0.39
CCNE1 P24864 4/20 0.39
CDK2 P24941 4/20 0.39
ROCK1 Q13464 4/20 0.39
DBF4 Q9UBU7 4/20 0.39
HCAR2 Q8TDS4 1/20 0.38
TP53 P04637 1/20 0.37
CTSV O60911 1/20 0.36
CTSL P07711 1/20 0.36
CTSB P07858 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL37626 0.89 PDE5A (0.80) PDE5APDE9APDE1APDE1BPDE1C
SCHEMBL38035 0.87 PDE5A (0.55) PDE5AMAPTRAB9AKDM4ELMNA
SCHEMBL37798 0.85 PDE5A (1.00) PDE5APDE9APDE1APDE1BPDE1C
SCHEMBL38176 0.85 PDE5A (0.73) PDE5APDE9APDE1APDE1BPDE1C
SCHEMBL37864 0.84 PDE5A (0.82) PDE5APDE9APDE1APDE1BPDE1C
SCHEMBL46289 0.80 PDE5A (0.76) PDE5APDE9APDE1APDE1BPDE1C
SCHEMBL38098 0.78 PDE5A (0.56) PDE5APDE9APDE1APDE1BPDE1C
SCHEMBL38275 0.78 PDE5A (0.69) PDE5APDE9APDE1APDE1BPDE1C
SCHEMBL38312 0.77 PDE5A (0.70) PDE5APDE9APDE1APDE1BPDE1C
SCHEMBL38180 0.76 PDE5A (0.60) PDE5AMAPTRAB9AKDM4ELMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012004900-A1 THIENOPYRIMIDINE COMPOUNDS ASKA PHARMACEUTICAL CO., LTD. (JP) 2012-01-12 WO disclosed