SCHEMBL386730

SCHEMBL386730

[CH2]C[Si](C)(c1ccccc1)c1ccccc1

nearest known ligand 0.39

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.39
ESR2 Q92731 1/20 0.39
MAPT P10636 1/20 0.35
NR1H2 P55055 2/20 0.32
NR1H3 Q13133 2/20 0.32
TP53 P04637 1/20 0.32
BRD4 O60885 1/20 0.31
BRD2 P25440 1/20 0.31
TSHR P16473 2/20 0.31
LMNA P02545 1/20 0.30
ALOX12 P18054 1/20 0.30
ACHE P22303 1/20 0.30
PTGS1 P23219 1/20 0.30
PTGS2 P35354 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL940805 0.79 MAPT (0.44) ESR1ESR2MAPTNR1H2NR1H3
SCHEMBL1270651 0.78 ESR1 (0.42) ESR1ESR2MAPTNR1H2NR1H3
SCHEMBL9225762 0.78 ESR1 (0.42) ESR1ESR2MAPTNR1H2NR1H3
SCHEMBL12191013 0.76 ESR1 (0.41) ESR1ESR2MAPTNR1H2NR1H3
SCHEMBL4908749 0.75 ESR1 (0.33) ESR1ESR2MAPT
SCHEMBL9339400 0.74 ESR1 (0.39) ESR1ESR2MAPTNR1H2NR1H3
SCHEMBL7935088 0.74 ESR1 (0.44) ESR1ESR2MAPTNR1H2NR1H3
SCHEMBL10427763 0.74 NR1H2 (0.41) ESR1ESR2MAPTNR1H2NR1H3
SCHEMBL1270667 0.74 ESR1 (0.39) ESR1ESR2MAPTNR1H2NR1H3
SCHEMBL7517705 0.74 ESR1 (0.39) ESR1ESR2MAPTNR1H2NR1H3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 233 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3643706-B1 MODIFIED NUCLEIC ACID MONOMERS AND OLIGONUCLEIC ACID ANALOGUES, WITH HIGH BIOLOGICAL STABILITY AND TARGET GENE SILENCING ACTIVITY, FOR USE IN THERAPY AND DIAGNOSIS OF CANCER AND VIRAL DISEASES EISAI R&D MAN CO LTD (JP) 2023-11-15 EP claimed
EP-2921499-B1 METHOD FOR LIQUID-PHASE SYNTHESIS OF NUCLEIC ACIDS TAKEDA PHARMACEUTICALS CO (JP) 2020-01-22 EP claimed
US-9896473-B2 Thiol compounds and the use thereof for the synthesis of modified oligonucleotides ETABLISSEMENT FRANCAIS DU SANG (FR) 2018-02-20 US claimed
US-9714560-B2 Protected scale inhibitors and methods relating thereto HALLIBURTON ENERGY SERVICES, INC. (US) 2017-07-25 US claimed
EP-2834253-B1 THIOL COMPOUNDS AND THE USE THEREOF FOR THE SYNTHESIS OF MODIFIED OLIGONUCLEOTIDES CENTRE NAT DE LA RECH SCIENT (C N R S ) (FR) 2017-03-29 EP claimed
US-20150158964-A1 THIOL COMPOUNDS AND THE USE THEREOF FOR THE SYNTHESIS OF MODIFIED OLIGONUCLEOTIDES UNIVERSITE CLAUDE BERNARD LYON 1 (FR) 2015-06-11 US claimed
US-20100323000-A1 METHOD AND PROCESS FOR PREPARING CARDIOLIPIN NEOPHARM, INC. (US) 2010-12-23 US claimed
EP-2088865-A2 GUGGULPHOSPHOLIPID METHODS AND COMPOSITIONS Jina Pharmaceuticals Inc. (US) 2009-08-19 EP claimed
WO-2008058156-A9 GUGGULPHOSPHOLIPID METHODS AND COMPOSITIONS JINA PHARMACEUTICALS INC (US) 2008-12-04 WO claimed
EP-1986607-A2 METHOD AND PROCESS FOR PREPARING CARDIOLIPIN Neopharm, Inc. (US) 2008-11-05 EP claimed
US-6172217-B1 SULFURIZATION OF PHOSPORDIAMIDITE; DEBLOCKING ISIS PHARMACEUTICALS INC. 2001-01-09 US claimed
US-6103891-A Method for the synthesis of nucleotide or oligonucleotide phosphoramidites ISIS PHARMACEUTICALS, INC. (US) 2000-08-15 US claimed
EP-0948512-A1 METHOD OF SYNTHESIZING PHOSPHOROTHIOATE OLIGONUCLEOTIDES ISIS PHARMACEUTICALS, INC. (US) 1999-10-13 EP claimed
EP-0948514-A1 METHOD FOR THE SYNTHESIS OF NUCLEOTIDE OR OLIGONUCLEOTIDE PHOSPHORAMIDITES ISIS PHARMACEUTICALS, INC. (US) 1999-10-13 EP claimed
US-5955600-A Method for the synthesis of nucleotide or oligonucleotide phosphoramidites ISIS PHARMACEUTICALS, INC. (US) 1999-09-21 US claimed
WO-1998029427-A1 METHOD OF SYNTHESIZING PHOSPHOROTHIOATE OLIGONUCLEOTIDES ISIS PHARMACEUTICALS, INC. (US) 1998-07-09 WO claimed
WO-1998029429-A1 METHOD FOR THE SYNTHESIS OF NUCLEOTIDE OR OLIGONUCLEOTIDE PHOSPHORAMIDITES ISIS PHARMACEUTICALS, INC. (US) 1998-07-09 WO claimed
US-5721350-A Deuterated nucleosides CHATTOPADHYAYA JYOTI (SE) 1998-02-24 US claimed
EP-0648220-A1 DEUTERATED NUCLEOSIDES CHATTOPADHYAYA, Jyoti (SE) 1995-04-19 EP claimed
WO-1993025566-A1 DEUTERATED NUCLEOSIDES CHATTOPADHYAYA JYOTI (SE) 1993-12-23 WO claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150158964-A1 THIOL COMPOUNDS AND THE USE THEREOF FOR THE SYNTHESIS OF MODIFIED OLIGONUCLEOTIDES TST, APEX1, TMT1A ESR1 4596/4885ESR2 4257/4885MAPT 1441/4885
US-20100323000-A1 METHOD AND PROCESS FOR PREPARING CARDIOLIPIN PHOSPHO1, SGMS1, SGMS2 ESR1 4835/4885ESR2 4861/4885MAPT 4674/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.