SCHEMBL3874013

SCHEMBL3874013

O=CC(Br)c1cc(OCc2ccccc2)c(OCc2ccccc2)c([N+](=O)[O-])c1

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 1/20 0.44
ADRA1D P25100 1/20 0.44
ADRA1A P35348 1/20 0.44
ADRA1B P35368 1/20 0.44
CTSV O60911 4/20 0.43
CTSL P07711 4/20 0.43
PIN1 Q13526 2/20 0.41
POLB P06746 1/20 0.41
PTGES O14684 1/20 0.41
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
MAPT P10636 1/20 0.40
CYP19A1 P11511 3/20 0.40
SGMS2 Q8NHU3 1/20 0.40
CYP11B1 P15538 1/20 0.38
CYP11B2 P19099 1/20 0.38
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21199371 0.86 CCNB2 (0.43) HTR1AADRA1DADRA1AADRA1BPOLB
SCHEMBL4286871 0.86 POLB (0.50) HTR1AADRA1DADRA1AADRA1BCTSV
SCHEMBL8077523 0.77 CYP19A1 (0.55) HTR1AADRA1DADRA1AADRA1BCTSV
SCHEMBL3874634 0.76 MEN1 (0.39) HTR1AADRA1DADRA1AADRA1BCTSV
SCHEMBL10477773 0.76 L3MBTL1 (0.43) POLBMEN1KMT2AMAPTNPC1
SCHEMBL4947751 0.75 MEN1 (0.42) HTR1AADRA1DADRA1AADRA1BCTSV
SCHEMBL27468143 0.74 POLB (0.48) HTR1AADRA1DADRA1AADRA1BCTSV
SCHEMBL1447206 0.74 CTSV (0.55) CTSVCTSLPOLBPTGESMEN1
SCHEMBL1447138 0.73 SGMS2 (0.47) HTR1AADRA1DADRA1AADRA1BCTSV
SCHEMBL3875000 0.73 ALDH1A1 (0.45) MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2027091-A1 NEW PHARMACEUTICAL COMPOUNDS BIAL - Portela & Ca., S.A. (PT) 2009-02-25 EP disclosed
EP-1907382-A1 NITROCATECHOL DERIVATIVES AS COMT INHIBITORS Portela & C.A. S.A (PT) 2008-04-09 EP disclosed
WO-2007117165-A1 NEW PHARMACEUTICAL COMPOUNDS BIAL - PORTELA & CA, S.A. (PT) 2007-10-18 WO disclosed
WO-2007013830-A1 NITROCATECHOL DERIVATIVES AS COMT INHIBITORS PORTELA & CA. S.A. (PT) 2007-02-01 WO disclosed