SCHEMBL3882575

SCHEMBL3882575

CC(Cc1cc(N)c(OC2CCCCC2)c(-c2ccc3[nH]ccc3c2)c1)C(=O)O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 1/20 0.43
APP P05067 1/20 0.37
EPHX1 P07099 1/20 0.36
AR P10275 1/20 0.35
ENPP2 Q13822 1/20 0.35
C5AR1 P21730 1/20 0.34
THRA P10827 1/20 0.34
THRB P10828 1/20 0.34
SMYD3 Q9H7B4 1/20 0.34
PARP10 Q53GL7 1/20 0.33
PARP11 Q9NR21 1/20 0.33
CHRNB2 P17787 1/20 0.33
CHRNB4 P30926 1/20 0.33
CHRNA3 P32297 1/20 0.33
CHRNA7 P36544 1/20 0.33
CHRNA4 P43681 1/20 0.33
CHRNA10 Q9GZZ6 1/20 0.33
CHRNA9 Q9UGM1 1/20 0.33
MCL1 Q07820 1/20 0.33
MAP3K11 Q16584 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3882901 0.99 PTGS2 (0.43) PTGS2APPEPHX1ARENPP2
SCHEMBL3897348 0.88 PTGS2 (0.41) PTGS2APPARENPP2THRA
SCHEMBL3882470 0.88 PTGS2 (0.41) PTGS2ARENPP2SMYD3MET
SCHEMBL3884011 0.86 APP (0.41) PTGS2APPTHRATHRB
SCHEMBL3884624 0.86 PTGS2 (0.40) PTGS2APPEPHX1ENPP2C5AR1
SCHEMBL3882109 0.85 PTGS2 (0.41) PTGS2APPEPHX1ARENPP2
SCHEMBL3883630 0.85 THRA (0.50) PTGS2EPHX1ARENPP2THRA
SCHEMBL3883960 0.85 FFAR4 (0.39) PTGS2APP
SCHEMBL3883671 0.84 PTGS2 (0.43) PTGS2APPEPHX1ENPP2C5AR1
SCHEMBL3680532 0.84 THRA (0.48) PTGS2EPHX1ARENPP2THRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1477472-B1 SUBSTITUTED PHENYLALKANOIC ACID DERIVATIVE AND USE THEREOF ASAHI KASEI PHARMA CORP (JP) 2009-01-14 EP claimed