SCHEMBL3889593

SCHEMBL3889593

O=C1NCC(c2cccc(Cc3ccccc3)c2)N1c1ccc(CO)cc1F

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 4/20 0.36
S1PR3 Q99500 4/20 0.36
FEN1 P39748 1/20 0.36
CFTR P13569 1/20 0.35
IDH1 O75874 1/20 0.34
SLC5A2 P31639 1/20 0.34
P2RX7 Q99572 2/20 0.33
PARP11 Q9NR21 1/20 0.33
LTA4H P09960 1/20 0.32
CHRNB4 P30926 1/20 0.32
CHRNA3 P32297 1/20 0.32
KCNH2 Q12809 1/20 0.32
PDPK1 O15530 1/20 0.32
HDAC1 Q13547 1/20 0.32
HDAC8 Q9BY41 1/20 0.32
HDAC6 Q9UBN7 1/20 0.32
HDAC5 Q9UQL6 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3556370 0.70 CFTR (0.43) S1PR1S1PR3CFTRIDH1LTA4H
SCHEMBL3884188 0.65 QPCT (0.35) HDAC8
SCHEMBL4037907 0.63 QPCT (0.43)
SCHEMBL4430768 0.63 TSHR (0.59) CFTRIDH1SLC5A2
SCHEMBL1602448 0.62 S1PR1 (0.67) S1PR1S1PR3CFTRIDH1LTA4H
SCHEMBL4553559 0.61 QPCT (0.51) HDAC1HDAC8HDAC6HDAC5
SCHEMBL11576495 0.60 TSHR (0.52) IDH1LTA4HCHRNB4CHRNA3HDAC8
SCHEMBL1280879 0.59 LTC4S (0.53) HDAC1HDAC8HDAC6
SCHEMBL3362040 0.58 CALM1 (0.55) IDH1LTA4H
SCHEMBL9560915 0.58 BCL2 (0.47) CFTRIDH1SLC5A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2010524-A2 S1P RECEPTOR MODULATING COMPOUNDS Epix Delaware, Inc. (US) 2009-01-07 EP disclosed
WO-2007109330-A2 S1P RECEPTOR MODULATING COMPOUNDS EPIX DELAWARE, INC. (US) 2007-09-27 WO disclosed