SCHEMBL39065

SCHEMBL39065

CCOC(=O)c1cccnc1Nc1cc(OCCOC)cc(-c2cn3ncccc3n2)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 3/20 0.41
MEN1 O00255 4/20 0.37
KMT2A Q03164 4/20 0.37
MAPK1 P28482 2/20 0.37
PKM P14618 1/20 0.37
MAPT P10636 6/20 0.37
POLB P06746 2/20 0.36
ALDH1A1 P00352 2/20 0.36
MAP2K1 Q02750 1/20 0.36
AAK1 Q2M2I8 2/20 0.36
GAA P10253 1/20 0.36
KDR P35968 1/20 0.36
MAP4K4 O95819 1/20 0.35
EGFR P00533 2/20 0.35
ERBB2 P04626 2/20 0.35
MAP4K2 Q12851 1/20 0.35
NPC1 O15118 2/20 0.35
RAB9A P51151 2/20 0.35
NPSR1 Q6W5P4 1/20 0.35
NFKB1 P19838 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL44718 0.89 MAP4K2 (0.45) HTTMEN1KMT2AMAPK1PKM
SCHEMBL44934 0.85 AAK1 (0.46) HTTMEN1KMT2AMAPK1PKM
SCHEMBL44514 0.76 AAK1 (0.48) HTTMEN1KMT2AMAPK1PKM
SCHEMBL4167706 0.73 MEN1 (0.58) HTTMEN1KMT2AMAPK1PKM
SCHEMBL44171 0.73 ROCK1 (0.41)
SCHEMBL44007 0.73 ALDH1A1 (0.41) HTTMAPTPOLBALDH1A1NPC1
SCHEMBL44632 0.72 LMNA (0.36) MAPTPOLBLMNA
SCHEMBL44471 0.72 ROCK1 (0.40) MEN1KMT2AMAPTALDH1A1GAA
SCHEMBL43813 0.72 LMNA (0.54) HTTMEN1KMT2AMAPK1PKM
SCHEMBL45017 0.71 PIK3CA (0.35) PKMMAPTALDH1A1GAAKDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011137587-A1 CYTOKINE INHIBITORS HUTCHISON MEDIPHARMA LIMITED (CN) 2011-11-10 WO claimed
WO-2011137587-A1 CYTOKINE INHIBITORS HUTCHISON MEDIPHARMA LIMITED (CN) 2011-11-10 WO disclosed
WO-2011137587-A1 CYTOKINE INHIBITORS HUTCHISON MEDIPHARMA LIMITED (CN) 2011-11-10 WO disclosed