SCHEMBL3928007

SCHEMBL3928007

Nc1ccc2ccoc(=O)c2c1.O=c1ccnc2ccccn12

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 2/20 0.56
GRM5 P41594 3/20 0.38
PRKDC P78527 1/20 0.34
KDM4E B2RXH2 3/20 0.32
CDK4 P11802 1/20 0.32
CDK2 P24941 1/20 0.32
ADORA2A P29274 1/20 0.32
ADORA2B P29275 1/20 0.32
ADORA1 P30542 1/20 0.32
SMN1; SMN2 Q16637 3/20 0.32
KMT2A Q03164 2/20 0.32
ALDH1A1 P00352 1/20 0.32
GLA P06280 1/20 0.32
GAA P10253 1/20 0.32
NPC1 O15118 1/20 0.32
MAPK1 P28482 1/20 0.32
RAB9A P51151 1/20 0.32
PKM P14618 2/20 0.32
MAPT P10636 1/20 0.32
HPGD P15428 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL163828 0.76 NPC1 (0.42) ADORA3KDM4ESMN1; SMN2KMT2AALDH1A1
SCHEMBL174735 0.75 ADORA3 (1.00) ADORA3GRM5PRKDCKDM4EADORA2A
Hydrochloric Acid SCHEMBL5127992 0.73 ADORA3 (0.96) ADORA3GRM5PRKDCKDM4EADORA2A
Hydrochloric Acid SCHEMBL5129999 0.73 ADORA3 (0.96) ADORA3GRM5PRKDCKDM4EADORA2A
Hydrochloric Acid SCHEMBL10598992 0.73 ADORA3 (0.96) ADORA3GRM5PRKDCKDM4EADORA2A
Trifluoroacetic Acid SCHEMBL5132448 0.64 ADORA3 (0.73) ADORA3GRM5KDM4ECDK4CDK2
SCHEMBL13256676 0.64 KDM4E (0.67) ADORA3KDM4EADORA2AADORA2BADORA1
SCHEMBL20602860 0.64 ADORA3 (0.61) ADORA3GRM5PRKDCKDM4EADORA2A
SCHEMBL3326263 0.62 ADORA3 (0.71) ADORA3GRM5PRKDCKDM4EADORA2A
SCHEMBL862066 0.62 KDM4E (0.51) ADORA3GRM5PRKDCKDM4EADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7541465-B2 Substituted 2-aminoacetamides and the use thereof PURDUE NEUROSCIENCE COMPANY (US) 2009-06-02 US disclosed
US-20060217403-A1 Substituted 2-aminoacetamides and the use thereof PURDUE NEUROSCIENCE COMPANY 2006-09-28 US disclosed
US-6281211-B1 TREATING A DISORDER RESPONSIVE TO THE BLOCKADE OF SODIUM CHANNELS EURO-CELTIQUE S.A. (LU) 2001-08-28 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060217403-A1 Substituted 2-aminoacetamides and the use thereof SLC1A2, GAP43, SCN2A ADORA3 226/4885GRM5 354/4885PRKDC 3004/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.