SCHEMBL163828

SCHEMBL163828

Nc1ccc2ccoc(=O)c2c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.42
RAB9A P51151 2/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
MAPT P10636 1/20 0.42
GFER P55789 1/20 0.42
CTDSP1 Q9GZU7 1/20 0.41
KMT2A Q03164 2/20 0.41
MAPK1 P28482 1/20 0.41
TYMS P04818 1/20 0.40
TDP1 Q9NUW8 2/20 0.36
PSEN1 P49768 1/20 0.36
PSEN2 P49810 1/20 0.36
APH1B Q8WW43 1/20 0.36
NCSTN Q92542 1/20 0.36
APH1A Q96BI3 1/20 0.36
PSENEN Q9NZ42 1/20 0.36
DYRK1A Q13627 1/20 0.36
CYP3A4 P08684 3/20 0.35
HSD17B10 Q99714 3/20 0.35
ALDH1A1 P00352 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3928007 0.76 ADORA3 (0.56) NPC1RAB9ASMN1; SMN2MAPTKMT2A
SCHEMBL31443864 0.76 PLG (0.40) KMT2ATYMSDYRK1ACYP3A4HSD17B10
SCHEMBL28859085 0.76 TYMS (0.38) MAPK1TYMSCYP3A4HSD17B10MAOA
SCHEMBL78392 0.76 CHEK1 (0.43) KMT2ATYMSCYP3A4HSD17B10ALDH1A1
SCHEMBL29402125 0.72 CTDSP1 (0.58) NPC1RAB9ASMN1; SMN2MAPTGFER
SCHEMBL12774936 0.72 CTDSP1 (0.58) NPC1RAB9ASMN1; SMN2MAPTGFER
SCHEMBL30578891 0.72 KMT2A (0.46) NPC1RAB9ASMN1; SMN2MAPTGFER
SCHEMBL17114053 0.72 KDM4E (0.51) NPC1RAB9ASMN1; SMN2MAPTTYMS
SCHEMBL25407064 0.71 PTPN1 (0.43) KMT2AALDH1A1MAOAPARP1MEN1
Isocoumarin SCHEMBL76183 0.70 PTGES (0.47) NPC1RAB9ASMN1; SMN2KMT2ATDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 660 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1809601-B1 COMPOUNDS FOR ALZHEIMER'S DISEASE MANFREDI JOHN (US) 2014-09-10 EP claimed
CN-102869261-A Compounds and therapeutic uses thereof MYREXIS INC 2013-01-09 CN claimed
EP-2542086-A1 COMPOUNDS AND THERAPEUTIC USES THEREOF Myrexis, Inc. (US) 2013-01-09 EP claimed
WO-2011109441-A1 COMPOUNDS AND THERAPEUTIC USES THEREOF MYREXIS, INC. (US) 2011-09-09 WO claimed
WO-2006135383-A2 INDAZOLES MYRIAD GENETICS, INC. (US) 2006-12-21 WO claimed
US-7015328-B2 Substituted coumarins and quinolines and analogs as activators of caspases and inducers of apoptosis and the use thereof CYTOVIA, INC. (US) 2006-03-21 US claimed
EP-1351691-A4 SUBSTITUTED 2-ARYL-4-ARYLAMINOPYRIMIDINES AND ANALOGS AS ACTIVATORS OF CASPASES AND INDUCERS OF APOPTOSIS AND THE USE THEREOF CYTOVIA INC (US) 2005-06-22 EP claimed
US-20040097503-A1 Substituted 2-aryl-4-arylaminopyrimidines and analogs as activators of caspases and inducers of apoptosis and the use thereof CYTOVIA, INC. 2004-05-20 US claimed
EP-1021418-B1 SUBSTITUTED 2,3-BENZODIAZEPIN-4-ONES AND THE USE THEREOF EURO CELTIQUE SA (LU) 2004-05-19 EP claimed
EP-1351691-A1 SUBSTITUTED 2-ARYL-4-ARYLAMINOPYRIMIDINES AND ANALOGS AS ACTIVATORS OF CASPASES AND INDUCERS OF APOPTOSIS AND THE USE THEREOF Cytovia, Inc. (US) 2003-10-15 EP claimed
US-20030069239-A1 Substituted 2-aryl-4-arylaminopyrimidines and analogs as activators or caspases and inducers of apoptosis and the use thereof CYTOVIA, INC. 2003-04-10 US claimed
US-6479484-B1 SUBSTITUTED 2-AMINOACETAMIDES AND THE DISCOVERY THAT THESE COMPOUNDS ACT AS BLOCKERS OF SODIUM CHANNELS; PAIN RELIEVERS, TREATMENT OF ARRYTHMIA, LOCAL ANESTHETICS EURO-CELTIQUE S.A. (LU) 2002-11-12 US claimed
WO-2002047690-A1 SUBSTITUTED 2-ARYL-4-ARYLAMINOPYRIMIDINES AND ANALOGS AS ACTIVATORS OF CASPASES AND INDUCERS OF APOPTOSIS AND THE USE THEREOF CYTOVIA, INC. (US) 2002-06-20 WO claimed
US-20260138956-A1 NOVEL COMPOUNDS AND USES THEREOF RECURSION PHARMACEUTICALS INC (US) 2026-05-21 US disclosed
EP-4720067-A1 BICYCLIC HETEROARYLAMIDES HAVING GPR68 MODULATING ACTIVITY Recursion Pharmaceuticals, Inc. (US) 2026-04-08 EP disclosed
US-12492197-B2 3,5-disubstituted pyrazole compounds as kinase inhibitors and uses thereof Impact Therapeutics (Shanghai), Inc (CN) 2025-12-09 US disclosed
EP-0564552-A1 USE OF CALPAIN INHIBITORS IN THE INHIBITION AND TREATMENT OF NEURODEGENERATION CORTEX PHARMACEUTICALS, INC. (US) 1993-10-13 EP disclosed
WO-1992011850-A2 USE OF CALPAIN INHIBITORS IN THE INHIBITION AND TREATMENT OF NEURODEGENERATION CORTEX PHARMACEUTICALS, INC. (US) 1992-07-23 WO disclosed
US-5089633-A Protease inhibitors, antiinflammatory agents GEORGIA TECH RESEARCH CORPORATION (US) 1992-02-18 US disclosed
US-5089634-A Protease inhibitors, antiinflammatory agents, anticoagulants GEORGIA TECH RESEARCH CORPORATION (US) 1992-02-18 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20260138956-A1 NOVEL COMPOUNDS AND USES THEREOF SLC10A1, NR3C2, CYP2C8 NPC1 9/4885RAB9A 418/4885SMN1; SMN2 999/4885
US-12492197-B2 3,5-disubstituted pyrazole compounds as kinase inhibitors and uses thereof CHEK1, CHEK2, CCNK NPC1 3791/4885RAB9A 1443/4885SMN1; SMN2 4202/4885
US-20030069239-A1 Substituted 2-aryl-4-arylaminopyrimidines and analogs as activators or caspases and inducers of apoptosis and the use thereof API5, CASP2, APAF1 NPC1 2878/4885RAB9A 3348/4885SMN1; SMN2 3150/4885
US-20040097503-A1 Substituted 2-aryl-4-arylaminopyrimidines and analogs as activators of caspases and inducers of apoptosis and the use thereof API5, CASP2, APAF1 NPC1 3014/4885RAB9A 3420/4885SMN1; SMN2 3214/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.