SCHEMBL3935992

SCHEMBL3935992

O=C(O)N1CCNC(CNc2cccnc2)C1

nearest known ligand 0.47

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
GRIN2B Q13224 3/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2D6 P10635 1/20 0.47
CYP2C9 P11712 1/20 0.47
ADRB1 P08588 4/20 0.43
EPHX2 P34913 2/20 0.39
NPC1 O15118 1/20 0.38
PKM P14618 1/20 0.38
RAB9A P51151 1/20 0.38
CXCR4 P61073 1/20 0.38
LCK P06239 1/20 0.37
ITGB3 P05106 1/20 0.37
ITGA2B P08514 1/20 0.37
NAMPT P43490 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL780721 0.84 GPR119 (0.48) GRIN2BCYP3A4CYP2D6CYP2C9NAMPT
SCHEMBL14720234 0.80 GRIN2B (0.64) GRIN2BCYP3A4CYP2D6CYP2C9EPHX2
SCHEMBL3933150 0.78 GRIN2B (0.46) GRIN2BCYP2C9EPHX2NPC1PKM
SCHEMBL4294740 0.74 MAN1B1 (0.43) ADRB1PKMCXCR4
SCHEMBL3933047 0.74 GRIN2B (0.45) GRIN2BCYP3A4CYP2D6CYP2C9EPHX2
SCHEMBL28989369 0.74 CHRNB2 (0.50) GRIN2BCYP2D6CYP2C9
SCHEMBL14603115 0.73 CHRNB2 (0.49) CYP2D6CYP2C9
SCHEMBL14346591 0.72 ADRA2A (0.42) GRIN2BCYP3A4CYP2D6CYP2C9RAB9A
SCHEMBL5337404 0.71 FAAH (0.44) GRIN2BCYP2D6EPHX2CXCR4
SCHEMBL23013515 0.70 SIGLEC9 (0.57) GRIN2BCYP3A4CYP2D6CYP2C9EPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2044038-A2 NOVEL PIPERAZINES, PHARMACEUTICAL COMPOSITIONS AND METHODS OF USE THEREOF Cornerstone Therapeutics Inc. (US) 2009-04-08 EP disclosed
WO-2007146066-A2 NOVEL PIPERAZINES, PHARMACEUTICAL COMPOSITIONS AND METHODS OF USE THEREOF CRITICAL THERAPEUTICS, INC. (US) 2007-12-21 WO disclosed