SCHEMBL3942976

SCHEMBL3942976

CN(CC(O)c1cccc(O)c1)C(=O)Oc1cnc(NCc2ccccc2Cl)nc1-c1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CASR P41180 1/20 0.41
HDAC3 O15379 2/20 0.38
HDAC1 Q13547 1/20 0.36
HDAC2 Q92769 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
SLC16A3 O15427 4/20 0.36
SLC16A1 P53985 3/20 0.36
MCTS1 Q9ULC4 3/20 0.36
OPRK1 P41145 2/20 0.35
VNN1 O95497 1/20 0.35
ADORA1 P30542 2/20 0.33
ALOX5 P09917 1/20 0.33
MEN1 O00255 1/20 0.33
LMNA P02545 1/20 0.33
KMT2A Q03164 1/20 0.33
VCP P55072 1/20 0.33
TP53 P04637 1/20 0.33
GAA P10253 1/20 0.33
MAPT P10636 1/20 0.33
MAOB P27338 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3952000 0.89 SLC16A3 (0.40) CASRHDAC3HDAC1HDAC2SLC16A3
SCHEMBL3945243 0.85 FYN (0.39) HDAC3HDAC1HDAC2HDAC6SLC16A3
SCHEMBL3946482 0.82 ALOX5 (0.39) SLC16A3ALOX5MEN1LMNAKMT2A
SCHEMBL3944707 0.79 CCNE2 (0.39) CASRGAAMAPT
SCHEMBL3947316 0.79 CASR (0.41) CASRSLC16A3ALOX5MEN1LMNA
SCHEMBL3942439 0.78 ALOX5 (0.38) OPRK1ALOX5MEN1LMNAKMT2A
SCHEMBL1384031 0.76 CASR (0.53) CASRHDAC3HDAC1HDAC2HDAC6
SCHEMBL3948201 0.76 SLC6A2 (0.37) CASRSLC16A3ALOX5MEN1LMNA
SCHEMBL3951648 0.76 TSPO (0.37) CASROPRK1ALOX5TP53
SCHEMBL1386304 0.76 SLC16A3 (0.41) CASRHDAC3HDAC1HDAC2SLC16A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1718632-B1 PYRIMIDINE DERIVATIVES AS OREXIN RECEPTOR ANTAGONISTS SANOFI AVENTIS (FR) 2009-04-22 EP claimed