SCHEMBL3946482

SCHEMBL3946482

CN(CC(O)c1cccc(O)c1)C(=O)Oc1cnc(N(C)C)nc1-c1ccccc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 1/20 0.39
PDK1 Q15118 1/20 0.38
MKNK1 Q9BUB5 1/20 0.37
SLC16A3 O15427 1/20 0.36
LMNA P02545 3/20 0.36
MEN1 O00255 3/20 0.36
KMT2A Q03164 3/20 0.36
HIF1A Q16665 4/20 0.35
TSHR P16473 2/20 0.35
ADRB2 P07550 1/20 0.35
ADRB1 P08588 1/20 0.35
HTR1A P08908 1/20 0.35
ADRA2A P08913 1/20 0.35
ADRB3 P13945 1/20 0.35
ADRA2B P18089 1/20 0.35
ADRA2C P18825 1/20 0.35
NFKB1 P19838 1/20 0.35
DRD1 P21728 1/20 0.35
HTR7 P34969 1/20 0.35
ADRA1A P35348 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3947316 0.90 CASR (0.41) ALOX5PDK1MKNK1SLC16A3LMNA
SCHEMBL3941835 0.89 ALOX5 (0.46) ALOX5LMNAMEN1KMT2ATSHR
SCHEMBL3942439 0.88 ALOX5 (0.38) ALOX5MKNK1LMNAMEN1KMT2A
SCHEMBL3948201 0.87 SLC6A2 (0.37) ALOX5PDK1MKNK1SLC16A3LMNA
SCHEMBL3953649 0.87 CASR (0.35) ALOX5PDK1SLC16A3LMNAMEN1
SCHEMBL3944917 0.86 BACE1 (0.41) MEN1KMT2AADRB2ADRB1ADRB3
SCHEMBL3952000 0.86 SLC16A3 (0.40) ALOX5PDK1SLC16A3LMNAMEN1
SCHEMBL3951123 0.85 BACE1 (0.41) ALOX5MEN1KMT2ARAB9AKDM4E
SCHEMBL3951861 0.85 GRM4 (0.41) NFKB1RAB9AKDM4E
SCHEMBL3952248 0.84 BACE1 (0.40) ALOX5ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1718632-B1 PYRIMIDINE DERIVATIVES AS OREXIN RECEPTOR ANTAGONISTS SANOFI AVENTIS (FR) 2009-04-22 EP claimed