SCHEMBL3944328

SCHEMBL3944328

CNCC(O)c1ccc(C#N)cc1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 6/20 0.61
TDP1 Q9NUW8 5/20 0.61
HIF1A Q16665 5/20 0.61
BLM P54132 4/20 0.61
ALDH1A1 P00352 2/20 0.61
HTR1A P08908 2/20 0.61
THPO P40225 2/20 0.61
SMN1; SMN2 Q16637 2/20 0.61
NMUR2 Q9GZQ4 1/20 0.61
CYP2C9 P11712 1/20 0.61
TAAR1 Q96RJ0 1/20 0.61
ADRB2 P07550 5/20 0.51
ADRB1 P08588 4/20 0.51
ADRB3 P13945 4/20 0.51
TSHR P16473 4/20 0.51
MAPT P10636 3/20 0.51
ADRA2A P08913 3/20 0.51
ADRA2B P18089 3/20 0.51
ADRA2C P18825 3/20 0.51
HSD17B10 Q99714 3/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9647484 0.82 HIF1A (0.49) KDM4ETDP1HIF1ABLMALDH1A1
SCHEMBL6666064 0.80 HIF1A (0.61) KDM4ETDP1HIF1ABLMALDH1A1
SCHEMBL21285889 0.79 GRIA1 (0.56) KDM4ETDP1HIF1ABLMALDH1A1
SCHEMBL21286133 0.79 GRIA1 (0.56) KDM4ETDP1HIF1ABLMALDH1A1
SCHEMBL29335774 0.79 GRIA1 (0.56) KDM4ETDP1HIF1ABLMALDH1A1
SCHEMBL18245963 0.79 LMNA (0.54) KDM4EALDH1A1MAPTLOXL2GAA
SCHEMBL2249403 0.79 LMNA (0.54) KDM4EALDH1A1MAPTLOXL2GAA
SCHEMBL11980400 0.79 CA12 (0.43) KDM4EALDH1A1MAPTLOXL2GAA
SCHEMBL3944322 0.77 F2R (0.41) KDM4ETDP1HIF1ABLMALDH1A1
Oxedrine SCHEMBL17726874 0.76 KDM4E (1.00) KDM4ETDP1HIF1ABLMALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1718632-B1 PYRIMIDINE DERIVATIVES AS OREXIN RECEPTOR ANTAGONISTS SANOFI AVENTIS (FR) 2009-04-22 EP claimed
US-20040116464-A1 Aryl-ethanolamine derivatives as antiviral agents PHARMACIA & UPJOHN COMPANY 2004-06-17 US disclosed
WO-2004022568-A1 ARYL-ETHANOLAMINE DERIVATIVES AS ANTIVIRAL AGENTS PHARMACIA & UPJOHN COMPANY LLC (US) 2004-03-18 WO disclosed