SCHEMBL3944646

SCHEMBL3944646

CC1(C)OC(=O)C(C(=O)CCc2ccccc2C#N)C(=O)O1

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
FFAR1 O14842 1/20 0.37
SIRT2 Q8IXJ6 1/20 0.37
SIRT1 Q96EB6 1/20 0.37
BACE1 P56817 1/20 0.35
P2RX7 Q99572 2/20 0.35
ALDH1A1 P00352 3/20 0.34
RAB9A P51151 2/20 0.34
GALR3 O60755 1/20 0.34
KMT2A Q03164 1/20 0.34
BRD4 O60885 1/20 0.33
TSHR P16473 4/20 0.33
NPC1 O15118 1/20 0.33
CASP3 P42574 1/20 0.32
SENP8 Q96LD8 1/20 0.32
SENP7 Q9BQF6 1/20 0.32
SENP6 Q9GZR1 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
CYP19A1 P11511 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3943900 0.81 CASP3 (0.39) BACE1ALDH1A1RAB9ANPC1CASP3
SCHEMBL956763 0.81 BACE1 (0.40) BACE1ALDH1A1KMT2ACASP3
SCHEMBL3941852 0.79 MTNR1A (0.44) CASP3TDP1
SCHEMBL6365366 0.72 ALDH1A1 (0.50) FFAR1ALDH1A1RAB9AGALR3BRD4
SCHEMBL12290424 0.70 NPSR1 (0.41) BACE1ALDH1A1RAB9AKMT2ANPC1
SCHEMBL30740885 0.70 FFAR1 (0.62) FFAR1
SCHEMBL447652 0.70 FFAR1 (0.62) FFAR1
SCHEMBL5642127 0.69 BACE1 (0.42) FFAR1BACE1P2RX7ALDH1A1TSHR
SCHEMBL9869709 0.69 CASP3 (0.41) ALDH1A1KMT2ACASP3
SCHEMBL2410483 0.69 FFAR1 (0.47) FFAR1ALDH1A1RAB9AGALR3TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009020457-A2 CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2009-02-12 WO disclosed
WO-2009020457-A2 CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2009-02-12 WO disclosed