SCHEMBL3969490

SCHEMBL3969490

COc1ccc(OCCc2c(C)nc3ccc(N4CCCCC4)cc3c2-c2ccc(F)cc2)cc1

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.41
HRH3 Q9Y5N1 2/20 0.41
APP P05067 4/20 0.41
ALDH1A1 P00352 3/20 0.41
MAPT P10636 3/20 0.41
KDM4E B2RXH2 2/20 0.41
HPGD P15428 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
ESR1 P03372 2/20 0.41
PIK3CA P42336 1/20 0.40
ACP1 P24666 1/20 0.40
LMNA P02545 1/20 0.40
SMO Q99835 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3963734 0.92 DRD2 (0.45) KCNH2HRH3KDM4EPIK3CA
SCHEMBL3964828 0.92 KCNH2 (0.43) KCNH2HRH3ALDH1A1MAPTKDM4E
SCHEMBL3966727 0.90 PIK3CD (0.40) KCNH2HRH3KDM4ENPSR1PIK3CA
SCHEMBL4198373 0.90 KCNH2 (0.39) KCNH2HRH3
SCHEMBL3970649 0.89 KCNH2 (0.41) KCNH2HRH3ESR1
SCHEMBL3962203 0.86 ELOVL1 (0.39) KCNH2HRH3MAPTLMNASMO
SCHEMBL3970363 0.86 DHFR (0.38) KCNH2HRH3MAPTPIK3CASMO
SCHEMBL3970650 0.85 ELOVL1 (0.36) KCNH2HRH3MAPTSMO
SCHEMBL3970359 0.84 ELOVL1 (0.46) KCNH2HRH3MAPTKDM4ELMNA
SCHEMBL3962208 0.84 HTR2A (0.47) HRH3ALDH1A1MAPTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009041904-A1 QUINOLINE COMPOUNDS HAVING AN ACTIVITY AGAINST THE GABAB RECEPTOR ASTRAZENECA AB (SE) 2009-04-02 WO claimed
WO-2009041904-A1 QUINOLINE COMPOUNDS HAVING AN ACTIVITY AGAINST THE GABAB RECEPTOR ASTRAZENECA AB (SE) 2009-04-02 WO disclosed