SCHEMBL3970650

SCHEMBL3970650

Cc1nc2ccc(N3CCCCC3)cc2c(-c2ccc(F)cc2)c1CCOc1cccc(N(C)C)c1

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ELOVL1 Q9BW60 1/20 0.36
IDO1 P14902 1/20 0.35
TDO2 P48775 1/20 0.35
IDO2 Q6ZQW0 1/20 0.35
SMO Q99835 1/20 0.35
KCNH2 Q12809 1/20 0.35
HRH3 Q9Y5N1 1/20 0.35
CCKAR P32238 2/20 0.34
MAPT P10636 4/20 0.33
MEN1 O00255 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C19 P33261 1/20 0.33
KMT2A Q03164 1/20 0.33
ADORA2A P29274 1/20 0.33
ADORA1 P30542 1/20 0.33
SLC6A2 P23975 1/20 0.33
SLC6A4 P31645 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3970363 0.86 DHFR (0.38) ELOVL1IDO1TDO2IDO2SMO
SCHEMBL3962203 0.85 ELOVL1 (0.39) ELOVL1IDO1TDO2IDO2SMO
SCHEMBL3970169 0.85 MAPK14 (0.41) CCKARMAPTMEN1CYP3A4CYP2D6
SCHEMBL3969490 0.85 KCNH2 (0.41) SMOKCNH2HRH3MAPT
SCHEMBL3963734 0.84 DRD2 (0.45) ELOVL1IDO1TDO2IDO2KCNH2
SCHEMBL3964828 0.84 KCNH2 (0.43) ELOVL1IDO1TDO2IDO2KCNH2
SCHEMBL4198373 0.83 KCNH2 (0.39) ELOVL1KCNH2HRH3
SCHEMBL3966727 0.82 PIK3CD (0.40) ELOVL1IDO1TDO2IDO2KCNH2
SCHEMBL3966950 0.82 IDO1 (0.35) IDO1TDO2IDO2SMOMAPT
SCHEMBL3970359 0.81 ELOVL1 (0.46) ELOVL1IDO1TDO2IDO2KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009041904-A1 QUINOLINE COMPOUNDS HAVING AN ACTIVITY AGAINST THE GABAB RECEPTOR ASTRAZENECA AB (SE) 2009-04-02 WO disclosed