SCHEMBL3969854

SCHEMBL3969854

COc1ccc(OCC(=O)NCCc2cn(-c3ccccc3)c3ccc(C(=O)O)cc23)cc1

nearest known ligand 0.66

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 3/20 0.66
MTNR1B P49286 3/20 0.66
PLA2G4A P47712 8/20 0.54
PTPN1 P18031 1/20 0.53
HTR6 P50406 1/20 0.50
CYP1A2 P05177 1/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2C19 P33261 1/20 0.46
HSD17B10 Q99714 1/20 0.46
NQO2 P16083 1/20 0.45
TDP1 Q9NUW8 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
ROCK1 Q13464 1/20 0.45
FAAH O00519 1/20 0.45
ACHE P22303 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4207303 0.93 MTNR1A (0.64) MTNR1AMTNR1BPLA2G4APTPN1HTR6
SCHEMBL3970925 0.90 MTNR1A (0.55) MTNR1AMTNR1BPLA2G4APTPN1HTR6
SCHEMBL3972866 0.90 MTNR1A (0.55) MTNR1AMTNR1BPLA2G4APTPN1CYP2C19
SCHEMBL13883746 0.88 MTNR1A (0.52) MTNR1AMTNR1BPLA2G4APTPN1CYP1A2
SCHEMBL3970852 0.87 MTNR1A (0.54) MTNR1AMTNR1BPLA2G4A
SCHEMBL13883771 0.85 MTNR1A (0.56) MTNR1AMTNR1BPLA2G4APTPN1HTR6
SCHEMBL3970351 0.76 MTNR1A (0.51) MTNR1AMTNR1BPLA2G4A
SCHEMBL3974599 0.75 PLA2G4A (0.54) MTNR1AMTNR1BPLA2G4AL3MBTL1
SCHEMBL13884082 0.73 MTNR1A (0.57) MTNR1AMTNR1BPLA2G4AHTR6NQO2
SCHEMBL3969848 0.73 PLA2G4A (0.52) MTNR1AMTNR1BPLA2G4AL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009047240-A1 INDOLE DERIVATIVES USEFUL AS PPAR ACTIVATORS SMITHKLINE BEECHAM CORPORATION (US) 2009-04-16 WO claimed
WO-2009047240-A1 INDOLE DERIVATIVES USEFUL AS PPAR ACTIVATORS SMITHKLINE BEECHAM CORPORATION (US) 2009-04-16 WO disclosed