SCHEMBL3971706

SCHEMBL3971706

CCOc1cc(CN(c2cc(C(F)(F)F)c(C(N)=O)cn2)C2CCNCC2)cc(OCC)c1F

nearest known ligand 0.35

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 7/20 0.35
SLC6A4 P31645 7/20 0.35
HTR2A P28223 3/20 0.35
TACR1 P25103 2/20 0.35
FLT4 P35916 1/20 0.34
PTK2 Q05397 1/20 0.34
SLC6A3 Q01959 2/20 0.34
KCNH2 Q12809 2/20 0.33
CHEK1 O14757 1/20 0.33
JAK2 O60674 1/20 0.33
NEK2 P51955 1/20 0.33
SSTR5 P35346 2/20 0.33
SCN9A Q15858 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3972620 0.88 TACR1 (0.38) SLC6A2SLC6A4TACR1FLT4PTK2
SCHEMBL3973958 0.85 SSTR5 (0.40) SLC6A2SLC6A4HTR2ATACR1FLT4
SCHEMBL3979706 0.82 REN (0.44) SLC6A2SLC6A4TACR1FLT4PTK2
SCHEMBL3974580 0.82 REN (0.41) SLC6A2SLC6A4HTR2ATACR1FLT4
SCHEMBL3977756 0.81 REN (0.41) HTR2ATACR1FLT4PTK2
SCHEMBL3972445 0.81 SSTR5 (0.40) SLC6A2SLC6A4HTR2ATACR1FLT4
SCHEMBL3968591 0.81 GAA (0.38) SLC6A2SLC6A4HTR2ATACR1SLC6A3
SCHEMBL3973837 0.81 REN (0.40) SLC6A2SLC6A4HTR2AFLT4PTK2
SCHEMBL3978560 0.80 RXRA (0.42) SSTR5
SCHEMBL3970028 0.80 ALDH1A1 (0.37) SLC6A2SLC6A4HTR2ATACR1SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2054385-A2 PHENYL, PYRIDINE AND QUINOLINE DERIVATIVES F. Hoffmann-Roche AG (CH) 2009-05-06 EP claimed
WO-2008019967-A2 PHENYL, PYRIDINE AND QUINOLINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2008-02-21 WO claimed
EP-2054385-A2 PHENYL, PYRIDINE AND QUINOLINE DERIVATIVES F. Hoffmann-Roche AG (CH) 2009-05-06 EP disclosed
WO-2008019967-A2 PHENYL, PYRIDINE AND QUINOLINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2008-02-21 WO disclosed