SCHEMBL3970028

SCHEMBL3970028

CCOc1cc(CN(c2cc(C(F)(F)F)c(C(=O)OC)cn2)C2CCNCC2)ccc1O

nearest known ligand 0.37

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.37
HTT P42858 1/20 0.37
GAA P10253 3/20 0.37
SMN1; SMN2 Q16637 1/20 0.36
TACR1 P25103 3/20 0.36
MAPT P10636 1/20 0.35
LMNA P02545 1/20 0.35
TP53 P04637 1/20 0.35
TOP2A P11388 1/20 0.34
SLC6A2 P23975 5/20 0.34
SLC6A4 P31645 5/20 0.34
SLC6A3 Q01959 3/20 0.34
KCNH2 Q12809 1/20 0.34
HTR2A P28223 2/20 0.33
KDM4E B2RXH2 1/20 0.33
TDP1 Q9NUW8 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3977756 0.92 REN (0.41) ALDH1A1HTTSMN1; SMN2TACR1MAPT
SCHEMBL3968591 0.92 GAA (0.38) ALDH1A1GAATACR1LMNATP53
SCHEMBL3977946 0.91 MAPT (0.40) ALDH1A1HTTSMN1; SMN2TACR1MAPT
SCHEMBL3972591 0.85 REN (0.43) GAASMN1; SMN2TACR1LMNAKDM4E
SCHEMBL3974580 0.84 REN (0.41) ALDH1A1TACR1SLC6A2SLC6A4HTR2A
SCHEMBL3972940 0.84 ALOX15 (0.40) GAAMAPTSLC6A2SLC6A4HTR2A
SCHEMBL3970195 0.84 SLC6A2 (0.37) ALDH1A1HTTGAASMN1; SMN2TACR1
SCHEMBL3972620 0.82 TACR1 (0.38) TACR1SLC6A2SLC6A4SLC6A3KCNH2
SCHEMBL3973372 0.80 RXRA (0.41) ALDH1A1GAAMAPTSLC6A2SLC6A4
SCHEMBL3971706 0.80 SLC6A2 (0.35) TACR1SLC6A2SLC6A4SLC6A3KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2054385-A2 PHENYL, PYRIDINE AND QUINOLINE DERIVATIVES F. Hoffmann-Roche AG (CH) 2009-05-06 EP claimed
WO-2008019967-A2 PHENYL, PYRIDINE AND QUINOLINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2008-02-21 WO claimed
EP-2054385-A2 PHENYL, PYRIDINE AND QUINOLINE DERIVATIVES F. Hoffmann-Roche AG (CH) 2009-05-06 EP disclosed
WO-2008019967-A2 PHENYL, PYRIDINE AND QUINOLINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2008-02-21 WO disclosed