SCHEMBL3971708

SCHEMBL3971708

O=C(O)c1ccc2c(c1)c(CCCCN1CCc3cc(C(F)(F)F)ccc3C1)cn2-c1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 1/20 0.51
TNF P01375 2/20 0.43
TNFSF11 O14788 1/20 0.43
PLA2G4A P47712 1/20 0.41
KDM4E B2RXH2 1/20 0.41
ALOX15 P16050 1/20 0.41
APEX1 P27695 1/20 0.41
KMT2A Q03164 1/20 0.41
HSD17B10 Q99714 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
DRD2 P14416 5/20 0.40
DRD3 P35462 5/20 0.40
HTR1A P08908 3/20 0.39
HTR2A P28223 3/20 0.39
HTR7 P34969 3/20 0.39
HRH1 P35367 3/20 0.39
HTR2B P41595 3/20 0.39
SLC6A4 P31645 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3973169 0.85 ABCB1 (0.51) ABCB1PLA2G4AKDM4EALOX15APEX1
SCHEMBL13883895 0.78 ABCB1 (0.53) ABCB1PLA2G4ADRD2DRD3
SCHEMBL3972294 0.77 NAMPT (0.48) PLA2G4A
SCHEMBL1356475 0.72 TNF (0.51) TNFTNFSF11PLA2G4AKMT2A
SCHEMBL3971256 0.71 NPC1 (0.47) PLA2G4AKMT2A
SCHEMBL31378117 0.71 TEAD1 (0.55) PLA2G4AKDM4E
SCHEMBL14489662 0.70 SIGMAR1 (0.56)
SCHEMBL7962844 0.69 ACACB (0.45) ABCB1DRD2DRD3HTR1AHTR2A
SCHEMBL13883789 0.69 MTNR1A (0.45) PLA2G4A
SCHEMBL1357522 0.69 TNF (0.48) TNFTNFSF11PLA2G4AKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009047240-A1 INDOLE DERIVATIVES USEFUL AS PPAR ACTIVATORS SMITHKLINE BEECHAM CORPORATION (US) 2009-04-16 WO disclosed