SCHEMBL3972294

SCHEMBL3972294

O=C(O)c1ccc2c(c1)c(CCCCNC(=O)c1ccc(C(F)(F)F)cc1)cn2-c1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 3/20 0.48
PLA2G4A P47712 4/20 0.46
MTNR1A P48039 1/20 0.46
MTNR1B P49286 1/20 0.46
MLYCD O95822 1/20 0.45
HDAC1 Q13547 2/20 0.44
HDAC2 Q92769 1/20 0.44
HDAC3 O15379 1/20 0.44
SIGMAR1 Q99720 2/20 0.44
TMEM97 Q5BJF2 1/20 0.44
TRPV1 Q8NER1 1/20 0.44
SLC6A5 Q9Y345 1/20 0.43
P2RY14 Q15391 2/20 0.42
OPRD1 P41143 1/20 0.42
RORC P51449 1/20 0.41
EPHX2 P34913 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3971256 0.91 NPC1 (0.47) PLA2G4AMTNR1AMTNR1BHDAC1HDAC2
SCHEMBL3976494 0.87 NPC1 (0.52) PLA2G4AMTNR1AMTNR1BHDAC1HDAC2
SCHEMBL13883789 0.83 MTNR1A (0.45) PLA2G4AMTNR1AMTNR1BRORCEPHX2
SCHEMBL3976741 0.83 MTNR1A (0.49) PLA2G4AMTNR1AMTNR1BHDAC1HDAC2
SCHEMBL3971346 0.81 NPC1 (0.44) PLA2G4AHDAC1HDAC2
SCHEMBL31378117 0.78 TEAD1 (0.55) PLA2G4ARORC
SCHEMBL3971708 0.77 ABCB1 (0.51) PLA2G4A
SCHEMBL13883740 0.76 NPC1 (0.48) PLA2G4AMTNR1AMTNR1BHDAC1HDAC2
SCHEMBL3971172 0.75 PTAFR (0.48) HDAC3
SCHEMBL1356475 0.74 TNF (0.51) PLA2G4ARORC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009047240-A1 INDOLE DERIVATIVES USEFUL AS PPAR ACTIVATORS SMITHKLINE BEECHAM CORPORATION (US) 2009-04-16 WO disclosed
WO-2009047240-A1 INDOLE DERIVATIVES USEFUL AS PPAR ACTIVATORS SMITHKLINE BEECHAM CORPORATION (US) 2009-04-16 WO disclosed