SCHEMBL3986985

SCHEMBL3986985

COc1ccc2c(c1)c(C(=O)c1cc(Cl)ncn1)cn2C

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCG2 Q9UNQ0 1/20 0.47
MTNR1A P48039 8/20 0.42
MTNR1B P49286 8/20 0.42
NQO2 P16083 1/20 0.42
ADRB2 P07550 1/20 0.40
ALDH1A1 P00352 2/20 0.39
KDM4E B2RXH2 1/20 0.39
LMNA P02545 1/20 0.39
GLA P06280 1/20 0.39
GAA P10253 1/20 0.39
HPGD P15428 1/20 0.39
MAPK1 P28482 1/20 0.39
HTT P42858 1/20 0.39
HSD17B10 Q99714 1/20 0.39
RXFP1 Q9HBX9 1/20 0.39
NR4A2 P43354 1/20 0.39
JAK2 O60674 1/20 0.39
LCK P06239 1/20 0.39
IGF1R P08069 1/20 0.39
GSK3A P49840 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3995936 0.93 ALDH1A1 (0.44) ABCG2MTNR1AMTNR1BNQO2ALDH1A1
SCHEMBL3989840 0.89 MTNR1A (0.39) ABCG2MTNR1AMTNR1BNQO2NR4A2
SCHEMBL3996013 0.86 KDR (0.41) ALDH1A1KDM4ELMNAHSD17B10NR4A2
SCHEMBL3973248 0.84 KDM4E (0.42) ALDH1A1KDM4ENR4A2JAK2LCK
SCHEMBL3990318 0.83 NR4A2 (0.35) ABCG2MTNR1AMTNR1BALDH1A1KDM4E
SCHEMBL3972624 0.82 POLB (0.55) ALDH1A1LMNAHTTNR4A2RAB9A
SCHEMBL16312903 0.81 ABCG2 (0.61) ABCG2MTNR1AMTNR1BNQO2ADRB2
SCHEMBL3992947 0.79 POLB (0.38) ALDH1A1KDM4ELMNA
SCHEMBL3992240 0.79 POLB (0.38) ALDH1A1LMNAHTTNR4A2
SCHEMBL3978572 0.77 PCSK9 (0.40) ALDH1A1KDM4ELMNAHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2065382-A1 CGRP antagonists Boehringer Ingelheim Pharma GmbH & Co. KG (DE) 2009-06-03 EP disclosed