SCHEMBL3989840

SCHEMBL3989840

COC(=O)Oc1ccc2c(c1)c(C(=O)c1cc(Cl)ncn1)cn2C

nearest known ligand 0.39

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 9/20 0.39
MTNR1B P49286 9/20 0.39
NR4A2 P43354 8/20 0.39
ABCG2 Q9UNQ0 1/20 0.38
NQO2 P16083 1/20 0.38
CA12 O43570 1/20 0.35
CA9 Q16790 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3990318 0.94 NR4A2 (0.35) MTNR1AMTNR1BNR4A2ABCG2
SCHEMBL3986985 0.89 ABCG2 (0.47) MTNR1AMTNR1BNR4A2ABCG2NQO2
SCHEMBL3995936 0.83 ALDH1A1 (0.44) MTNR1AMTNR1BABCG2NQO2
SCHEMBL3996013 0.82 KDR (0.41) NR4A2CA12CA9
SCHEMBL3973248 0.80 KDM4E (0.42) NR4A2CA12CA9
SCHEMBL3972624 0.79 POLB (0.55) NR4A2
SCHEMBL4257184 0.78 PCSK9 (0.36) NR4A2
SCHEMBL4259652 0.78 NR4A2 (0.34) NR4A2ABCG2
SCHEMBL3992240 0.75 POLB (0.38) NR4A2CA12CA9
SCHEMBL3992947 0.75 POLB (0.38)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2065382-A1 CGRP antagonists Boehringer Ingelheim Pharma GmbH & Co. KG (DE) 2009-06-03 EP disclosed