SCHEMBL3973766

SCHEMBL3973766

NC(=O)c1ccc(-c2cccc(O)c2)s1.NC(=O)c1ccc(-c2cccc(OCCCl)c2)s1

nearest known ligand 0.53

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HSD17B1 P14061 11/20 0.53
HSD17B2 P37059 11/20 0.53
HPGDS O60760 4/20 0.52
EPHX2 P34913 1/20 0.47
ESRRG P62508 3/20 0.46
IKBKB O14920 1/20 0.45
ESR1 P03372 2/20 0.45
ESR2 Q92731 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1784939 0.94 EPHX2 (0.52) HSD17B1HSD17B2HPGDSEPHX2IKBKB
SCHEMBL1784584 0.83 HPGDS (0.73) HSD17B1HSD17B2HPGDSEPHX2ESRRG
SCHEMBL1786187 0.81 IKBKB (0.59) HSD17B2EPHX2IKBKB
SCHEMBL5605133 0.79 EPHX2 (0.61) HSD17B1HSD17B2EPHX2IKBKB
SCHEMBL5613367 0.75 HDAC6 (0.71) HSD17B1HSD17B2EPHX2IKBKB
SCHEMBL12607746 0.75 EPHX2 (0.43) HSD17B1HSD17B2EPHX2ESRRGESR1
SCHEMBL12607745 0.74 HSD17B2 (0.49) HSD17B1HSD17B2HPGDSEPHX2IKBKB
SCHEMBL12607747 0.72 ALDH1A1 (0.45) HSD17B1HSD17B2EPHX2
SCHEMBL1789489 0.72 FAAH (0.50) EPHX2
SCHEMBL3021743 0.72 CHRNB2 (0.61)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2054383-A2 NOVEL COMPOUNDS AS ANTAGONISTS OR INVERSE AGONISTS AT OPIOID RECEPTORS SmithKline Beecham Corporation (US) 2009-05-06 EP disclosed
WO-2008021849-A2 NOVEL COMPOUNDS AS ANTAGONISTS OR INVERSE AGONISTS AT OPIOID RECEPTORS SMITHKLINE BEECHAM CORPORATION (US) 2008-02-21 WO disclosed