SCHEMBL3974103

SCHEMBL3974103

COc1ccc2[nH]cc(C(=O)c3cc(Cl)ncn3)c2c1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.57
MEN1 O00255 2/20 0.57
KMT2A Q03164 2/20 0.57
MAPT P10636 2/20 0.57
NPSR1 Q6W5P4 2/20 0.57
MITF O75030 1/20 0.57
RAB9A P51151 1/20 0.57
NR4A2 P43354 2/20 0.56
CPT1A P50416 1/20 0.52
ALDH1A1 P00352 2/20 0.49
CYP1A2 P05177 1/20 0.49
CYP2C9 P11712 1/20 0.49
CYP2C19 P33261 1/20 0.49
IMPDH2 P12268 1/20 0.47
IMPDH1 P20839 1/20 0.47
TUBB1 Q9H4B7 2/20 0.47
HTR4 Q13639 2/20 0.46
KDM4E B2RXH2 3/20 0.45
SMN1; SMN2 Q16637 2/20 0.45
TP53 P04637 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27908679 0.81 NR4A2 (0.77) LMNAMEN1KMT2AMAPTNPSR1
SCHEMBL3990192 0.80 GPR84 (0.58) MEN1KMT2AMAPTNPSR1RAB9A
SCHEMBL10172506 0.77 CPS1 (0.47) LMNAMEN1KMT2ARAB9AALDH1A1
SCHEMBL3986985 0.76 ABCG2 (0.47) LMNARAB9ANR4A2ALDH1A1KDM4E
SCHEMBL28386254 0.76 NPSR1 (0.74) LMNAMEN1KMT2AMAPTNPSR1
SCHEMBL11794897 0.76 LMNA (0.74) LMNAMEN1KMT2AMAPTNPSR1
SCHEMBL21449261 0.75 NR4A2 (0.57) LMNAMEN1KMT2AMAPTNPSR1
SCHEMBL592889 0.75 NR4A2 (0.77) LMNAMEN1KMT2AMAPTNPSR1
SCHEMBL13302221 0.75 NPSR1 (0.72) LMNAMEN1KMT2AMAPTNPSR1
SCHEMBL3990312 0.75 TDO2 (0.41) NR4A2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2065382-A1 CGRP antagonists Boehringer Ingelheim Pharma GmbH & Co. KG (DE) 2009-06-03 EP disclosed
WO-2009050235-A1 CGRP ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2009-04-23 WO disclosed
WO-2009050235-A1 CGRP ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2009-04-23 WO disclosed