SCHEMBL3974248

SCHEMBL3974248

Nc1ccc(-c2ccnc3ccccc23)cc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NCF1 P14598 1/20 0.55
AURKA O14965 1/20 0.54
TTK P33981 1/20 0.54
AURKB Q96GD4 1/20 0.54
INCENP Q9NQS7 1/20 0.54
ACVR1 Q04771 4/20 0.50
GRM4 Q14833 4/20 0.49
CA12 O43570 2/20 0.49
CA1 P00915 2/20 0.49
CA2 P00918 2/20 0.49
CA9 Q16790 2/20 0.49
HTR2B P41595 1/20 0.49
MTNR1A P48039 1/20 0.49
KCNH2 Q12809 1/20 0.49
PIK3CA P42336 1/20 0.49
CYP1A2 P05177 1/20 0.47
LOXL2 Q9Y4K0 1/20 0.47
TGFBR1 P36897 3/20 0.46
MAPK14 Q16539 1/20 0.46
KDM4E B2RXH2 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27737402 0.87 CA12 (0.63) NCF1AURKATTKAURKBINCENP
SCHEMBL12074333 0.85 PIK3CA (0.65) NCF1AURKATTKAURKBINCENP
SCHEMBL30439957 0.84 TGFBR1 (0.60) NCF1AURKATTKAURKBINCENP
SCHEMBL35327 0.84 TGFBR1 (0.60) NCF1AURKATTKAURKBINCENP
SCHEMBL17945617 0.82 CYP1A2 (0.57) NCF1AURKATTKAURKBINCENP
SCHEMBL12580359 0.82 PIK3CA (0.54) AURKATTKAURKBINCENPACVR1
SCHEMBL12580413 0.82 PIK3CA (0.54) AURKATTKAURKBINCENPACVR1
SCHEMBL18805529 0.81 GRM4 (0.62) NCF1AURKATTKAURKBINCENP
SCHEMBL19219069 0.81 PIK3CA (0.71) NCF1AURKATTKAURKBINCENP
SCHEMBL3974245 0.81 ACVR1 (0.50) NCF1AURKATTKAURKBINCENP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10259800-B2 Method of fluorination using iodonium ylides THE GENERAL HOSPITAL CORPORATION (US) 2019-04-16 US disclosed
US-10259800-B2 Method of fluorination using iodonium ylides THE GENERAL HOSPITAL CORPORATION (US) 2019-04-16 US disclosed
EP-3240057-A1 ORGANIC ELECTROLUMINESCENT ELEMENT Hodogaya Chemical Co., Ltd. (JP) 2017-11-01 EP disclosed
US-20170121300-A1 METHOD OF FLUORINATION USING IODONIUM YLIDES THE GENERAL HOSPITAL CORPORATION 2017-05-04 US disclosed
US-20170121300-A1 METHOD OF FLUORINATION USING IODONIUM YLIDES THE GENERAL HOSPITAL CORPORATION 2017-05-04 US disclosed
US-20170121300-A1 METHOD OF FLUORINATION USING IODONIUM YLIDES THE GENERAL HOSPITAL CORPORATION 2017-05-04 US disclosed
US-7595317-B2 Barbituric acid derivatives as inhibitors of TNF-α converting enzyme (TACE) and/or matrix metalloproteinases BRISTOL-MYERS SQUIBB COMPANY (US) 2009-09-29 US disclosed
US-7294624-B2 Osteoporosis; antiarthritic agents BRISTOL MYERS SQUIBB COMPANY (US) 2007-11-13 US disclosed
US-20070167451-A1 BARBITURIC ACID DERIVATIVES AS INHIBITORS OF TNF-alpha CONVERTING ENZYME (TACE) AND/OR MATRIX METALLOPROTEINASES DUAN JINGWU 2007-07-19 US disclosed
WO-2003053941-A2 BARBITURIC ACID DERIVATIVES AS INHIBITORS OF TNF-ALPHA CONVERTING ENZYME (TACE) AND/OR MATRIX METALLOPROTEINASES BRISTOL-MYERS SQUIBB COMPANY (US) 2003-07-03 WO disclosed
CN-1092769-A Cyclic urea derivatives, the method that contains the pharmaceutical composition of these compounds and prepare them THOMAE GMBH DR K (DE) 1994-09-28 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170121300-A1 METHOD OF FLUORINATION USING IODONIUM YLIDES FLI1, ABL1, PFAS NCF1 1987/4885AURKA 408/4885TTK 1780/4885
US-20070167451-A1 BARBITURIC ACID DERIVATIVES AS INHIBITORS OF TNF-alpha CONVERTING ENZYME (TACE) AND/OR MATRIX METALLOPROTEINASES TNF, MMP9, MMP3 NCF1 992/4885AURKA 3775/4885TTK 3152/4885
US-10259800-B2 Method of fluorination using iodonium ylides FLI1, ABL1, PFAS NCF1 1987/4885AURKA 408/4885TTK 1780/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.