SCHEMBL3980490

SCHEMBL3980490

CC(=O)NCc1ccc(-c2ccc(OCC3CCN(C(=O)O)CC3)cn2)cc1

nearest known ligand 0.51

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CYP4F2 P78329 10/20 0.51
CYP4A11 Q02928 10/20 0.51
GPR119 Q8TDV5 9/20 0.50
HDAC1 Q13547 1/20 0.47
GPR183 P32249 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3981571 0.89 CYP4F2 (0.48) CYP4F2CYP4A11GPR119
SCHEMBL14191024 0.88 GPR119 (0.66) CYP4F2CYP4A11GPR119HDAC1
SCHEMBL3983094 0.86 CYP4F2 (0.52) CYP4F2CYP4A11GPR119GPR183
SCHEMBL3987843 0.82 GPR119 (0.54) CYP4F2CYP4A11GPR119HDAC1
SCHEMBL3983401 0.82 GPR119 (0.49) CYP4F2CYP4A11GPR119GPR183
SCHEMBL3983586 0.82 GPR119 (0.56) CYP4F2CYP4A11GPR119HDAC1GPR183
SCHEMBL3986034 0.81 GPR119 (0.52) CYP4F2CYP4A11GPR119GPR183
SCHEMBL3980457 0.81 GPR119 (0.61) CYP4F2CYP4A11GPR119GPR183
SCHEMBL3983576 0.81 LTA4H (0.40) GPR119
SCHEMBL3982981 0.80 CYP4F2 (0.50) CYP4F2CYP4A11GPR119GPR183

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2059516-A1 PYRIDINE COMPOUNDS FOR TREATING GPR119 RELATED DISORDERS BIOVITRUM AB (publ) (SE) 2009-05-20 EP claimed
US-20080103123-A1 New compounds BIOVITRUM (SE) 2008-05-01 US claimed
WO-2008025798-A1 PYRIDINE COMPOUNDS FOR TREATING GPR119 RELATED DISORDERS BIOVITRUM AB (PUBL) (SE) 2008-03-06 WO claimed
EP-2059516-A1 PYRIDINE COMPOUNDS FOR TREATING GPR119 RELATED DISORDERS BIOVITRUM AB (publ) (SE) 2009-05-20 EP disclosed
US-20080103123-A1 New compounds BIOVITRUM (SE) 2008-05-01 US disclosed
WO-2008025798-A1 PYRIDINE COMPOUNDS FOR TREATING GPR119 RELATED DISORDERS BIOVITRUM AB (PUBL) (SE) 2008-03-06 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080103123-A1 New compounds GPR119, GPR139, GPR180 CYP4F2 674/4885CYP4A11 147/4885GPR119 1/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.