SCHEMBL3989902

SCHEMBL3989902

COc1ccc(F)c2c(OS(C)(=O)=O)nc(Cc3ccc(Cl)cc3)nc12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 2/20 0.43
ALDH1A1 P00352 2/20 0.39
KDM4E B2RXH2 1/20 0.39
HPGD P15428 1/20 0.39
MAPT P10636 4/20 0.36
TSHR P16473 2/20 0.36
MEN1 O00255 1/20 0.35
LMNA P02545 1/20 0.35
KMT2A Q03164 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
CYP3A4 P08684 1/20 0.34
PSEN1 P49768 1/20 0.34
PSEN2 P49810 1/20 0.34
APH1B Q8WW43 1/20 0.34
NCSTN Q92542 1/20 0.34
APH1A Q96BI3 1/20 0.34
PSENEN Q9NZ42 1/20 0.34
SCN9A Q15858 1/20 0.34
HTT P42858 1/20 0.33
P2RX3 P56373 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3980812 0.72 ALDH1A1 (0.44) MAPK1ALDH1A1KDM4EHPGDMAPT
SCHEMBL3985590 0.71 CCNE2 (0.47) MAPK1ALDH1A1HPGDMAPTTSHR
SCHEMBL3984739 0.69 LMNA (0.38) MAPK1ALDH1A1KDM4EHPGDMAPT
SCHEMBL4300214 0.66 MAPK1 (0.53) MAPK1ALDH1A1KDM4EHPGDMAPT
SCHEMBL3984193 0.64 MAPT (0.50) MAPK1ALDH1A1KDM4EHPGDMAPT
SCHEMBL25328584 0.63 ALDH1A1 (0.41) ALDH1A1KDM4EHPGDMAPTMEN1
SCHEMBL3980996 0.61 PTGDR2 (0.39) MAPK1ALDH1A1KDM4EMAPTTSHR
SCHEMBL14919774 0.61 PDE4D (0.38) MAPK1ALDH1A1KDM4EHPGDTSHR
SCHEMBL2871982 0.61 MAPT (0.57) ALDH1A1MAPTLMNAKMT2AL3MBTL1
SCHEMBL16680513 0.60 PPARG (0.46) MAPK1ALDH1A1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009060209-A1 6,6-FUSED BICYCLIC AROMATIC COMPOUNDS AND THEIR THERAPEUTI USE ARGENTA DISCOVERY LIMITED (GB) 2009-05-14 WO disclosed