SCHEMBL3980812

SCHEMBL3980812

COc1ccc(F)c2cnc(Cc3ccc(Cl)cc3)nc12

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.44
KDM4E B2RXH2 1/20 0.44
HPGD P15428 1/20 0.44
MAPT P10636 4/20 0.43
TSHR P16473 2/20 0.43
MAPK1 P28482 3/20 0.42
L3MBTL1 Q9Y468 3/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
CYP1A2 P05177 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
LMNA P02545 1/20 0.39
HTR2C P28335 1/20 0.39
HTR2B P41595 1/20 0.39
CYP17A1 P05093 1/20 0.36
PDE5A O76074 1/20 0.36
TNKS O95271 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3980996 0.85 PTGDR2 (0.39) ALDH1A1KDM4EMAPTTSHRMAPK1
SCHEMBL3983651 0.82 PTGDR2 (0.43) MAPTTSHRTDP1
SCHEMBL3983803 0.80 HTR2C (0.41) KDM4EHPGDMAPTMAPK1L3MBTL1
SCHEMBL3984193 0.79 MAPT (0.50) ALDH1A1KDM4EHPGDMAPTTSHR
SCHEMBL25328601 0.78 ALDH1A1 (0.45) ALDH1A1KDM4ETNKSTNKS2PARP2
SCHEMBL4300214 0.74 MAPK1 (0.53) ALDH1A1KDM4EHPGDMAPTTSHR
SCHEMBL3989902 0.72 MAPK1 (0.43) ALDH1A1KDM4EHPGDMAPTTSHR
SCHEMBL3985590 0.67 CCNE2 (0.47) ALDH1A1HPGDMAPTTSHRMAPK1
SCHEMBL3989921 0.66 LMNA (0.41) ALDH1A1KDM4EHPGDMAPTTSHR
SCHEMBL3985579 0.65 LMNA (0.44) ALDH1A1KDM4EHPGDMAPTTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009060209-A1 6,6-FUSED BICYCLIC AROMATIC COMPOUNDS AND THEIR THERAPEUTI USE ARGENTA DISCOVERY LIMITED (GB) 2009-05-14 WO disclosed