SCHEMBL400608

SCHEMBL400608

Cc1ccc(C(=O)O)c(-c2ccc(C(F)(F)F)cc2)n1

nearest known ligand 0.52

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NTRK1 P04629 1/20 0.52
NTRK2 Q16620 1/20 0.52
RXRA P19793 1/20 0.49
RXRB P28702 1/20 0.49
SORT1 Q99523 8/20 0.48
DHODH Q02127 3/20 0.47
PTPN1 P18031 1/20 0.44
CYP2C8 P10632 1/20 0.44
KDM4E B2RXH2 2/20 0.44
ALDH1A1 P00352 2/20 0.44
HPGD P15428 2/20 0.44
HSD17B10 Q99714 2/20 0.44
USP2 O75604 1/20 0.42
CYP2C19 P33261 1/20 0.42
PPARD Q03181 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL398066 0.84 NTRK1 (0.52) NTRK1NTRK2SORT1DHODHPTPN1
SCHEMBL5532405 0.80 ALDH1A1 (0.54) NTRK1DHODHKDM4EALDH1A1HSD17B10
SCHEMBL6491306 0.79 PTPN1 (0.46) NTRK1RXRARXRBSORT1DHODH
SCHEMBL9355817 0.78 GABRP (0.48) SORT1KDM4EALDH1A1
SCHEMBL1550372 0.76 SMN1; SMN2 (0.69) RXRARXRBSORT1CYP2C8KDM4E
SCHEMBL7822583 0.76 MAPK1 (0.46) RXRARXRBDHODHCYP2C8KDM4E
SCHEMBL4597570 0.76 KIF11 (0.42) NTRK1NTRK2PTPN1KDM4E
SCHEMBL2555332 0.75 MGLL (0.43) NTRK1NTRK2DHODHPTPN1KDM4E
SCHEMBL402418 0.75 TDP1 (0.46) DHODHPTPN1KDM4EALDH1A1HPGD
SCHEMBL4197626 0.74 TDP1 (0.61) DHODHKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8101774-B2 Ester derivatives and medicinal use thereof JAPAN TOBACCO INC. (JP) 2012-01-24 US disclosed
US-8101774-B2 Ester derivatives and medicinal use thereof JAPAN TOBACCO INC. (JP) 2012-01-24 US disclosed
US-8101774-B2 Ester derivatives and medicinal use thereof JAPAN TOBACCO INC. (JP) 2012-01-24 US disclosed
EP-1803452-A1 ESTER DERIVATIVE AND PHARMACEUTICAL USE THEREOF Japan Tobacco, Inc. (JP) 2007-07-04 EP disclosed
EP-1803452-A1 ESTER DERIVATIVE AND PHARMACEUTICAL USE THEREOF Japan Tobacco, Inc. (JP) 2007-07-04 EP disclosed
US-20060089392-A1 Ester derivatives and medicinal use thereof JAPAN TOBACCO INC. (JP) 2006-04-27 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060089392-A1 Ester derivatives and medicinal use thereof MTTP, CETP, LIPA NTRK1 3420/4885NTRK2 2775/4885RXRA 2068/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.