SCHEMBL4006629

SCHEMBL4006629

C=C(OCC)c1ncnc2c1c(-c1ccccc1Cl)cn2CC(=O)O

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 5/20 0.38
KDM4E B2RXH2 4/20 0.38
ALDH1A1 P00352 4/20 0.38
HPGD P15428 2/20 0.38
NPSR1 Q6W5P4 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
GPR119 Q8TDV5 1/20 0.36
TP53 P04637 3/20 0.36
POLB P06746 1/20 0.36
EGFR P00533 1/20 0.35
SRC P12931 1/20 0.35
KDR P35968 1/20 0.35
MEN1 O00255 3/20 0.35
KMT2A Q03164 3/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
CCR4 P51679 1/20 0.35
CNR1 P21554 2/20 0.34
CNR2 P34972 1/20 0.34
P2RX7 Q99572 1/20 0.33
MCL1 Q07820 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13769538 0.92 MAPT (0.38) MAPTKDM4EALDH1A1HPGDNPSR1
SCHEMBL4014280 0.84 EGLN1 (0.34) MAPTKDM4ENPSR1TP53POLB
SCHEMBL13769676 0.82 MAPT (0.39) MAPTKDM4EALDH1A1HPGDNPSR1
SCHEMBL4007097 0.80 ALOX15 (0.36) MAPTKDM4EALDH1A1HPGDNPSR1
SCHEMBL4007615 0.80 SRC (0.43) MAPTPOLBSRCMEN1KMT2A
SCHEMBL4008754 0.79 FLT4 (0.44) MAPTALDH1A1HPGDPOLBSRC
SCHEMBL13769532 0.79 PDE4B (0.41) MAPTKDM4EALDH1A1HPGDNPSR1
SCHEMBL13769671 0.77 SRC (0.45) MAPTKDM4EALDH1A1HPGDNPSR1
SCHEMBL4006132 0.77 P2RX7 (0.43) MAPTKDM4EALDH1A1POLBSRC
SCHEMBL13769525 0.77 MAPT (0.40) MAPTKDM4EALDH1A1HPGDNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009080682-A1 PYRROLO[2,3-D]PYRIMIDINE DERIVATIVES AS CGRP RECEPTOR ANTAGONISTS GLAXO GROUP LIMITED (GB) 2009-07-02 WO disclosed