SCHEMBL4014280

SCHEMBL4014280

CC(=O)c1ncnc2c1c(-c1ccccc1Cl)cn2CC(=O)O

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGLN1 Q9GZT9 2/20 0.34
KIF11 P52732 1/20 0.34
KDM4E B2RXH2 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
POLB P06746 1/20 0.34
MAPT P10636 1/20 0.34
CCR4 P51679 1/20 0.34
SRC P12931 2/20 0.34
PTGDR2 Q9Y5Y4 1/20 0.33
NOTUM Q6P988 1/20 0.33
MCL1 Q07820 2/20 0.33
IGF1R P08069 1/20 0.33
ADK P55263 1/20 0.33
TP53 P04637 1/20 0.33
EGLN3 Q9H6Z9 1/20 0.33
P2RX7 Q99572 1/20 0.32
MEN1 O00255 1/20 0.32
NR2F2 P24468 1/20 0.32
KMT2A Q03164 1/20 0.32
PTGS2 P35354 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4013000 0.91 CCR4 (0.39) POLBCCR4PTGDR2MCL1P2RX7
SCHEMBL13769676 0.86 MAPT (0.39) KDM4ENPSR1MAPTSRCTP53
SCHEMBL4007615 0.86 SRC (0.43) EGLN1POLBMAPTCCR4SRC
SCHEMBL4006629 0.84 MAPT (0.38) KDM4ENPSR1POLBMAPTCCR4
SCHEMBL4007097 0.84 ALOX15 (0.36) EGLN1KDM4ENPSR1POLBMAPT
SCHEMBL4008754 0.83 FLT4 (0.44) EGLN1POLBMAPTCCR4SRC
SCHEMBL4006132 0.83 P2RX7 (0.43) EGLN1KDM4EPOLBMAPTSRC
SCHEMBL13769690 0.81 STAT3 (0.38) EGLN1POLBMAPTSRCPTGDR2
SCHEMBL4005788 0.80 MAPT (0.43) KDM4EMAPTADKTP53
SCHEMBL4006053 0.79 LMNA (0.47) KDM4ENPSR1POLBMAPTTP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009080682-A1 PYRROLO[2,3-D]PYRIMIDINE DERIVATIVES AS CGRP RECEPTOR ANTAGONISTS GLAXO GROUP LIMITED (GB) 2009-07-02 WO disclosed