SCHEMBL4013700

SCHEMBL4013700

Cc1cccc(CCc2cc(N)n[nH]2)c1

nearest known ligand 0.50

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 1/20 0.50
DAO P14920 2/20 0.49
GPR84 Q9NQS5 1/20 0.47
NOS1 P29475 1/20 0.45
NOS2 P35228 1/20 0.45
ALDH1A1 P00352 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
MPO P05164 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.42
IDO1 P14902 2/20 0.41
NPC1 O15118 1/20 0.41
MAPT P10636 1/20 0.41
RAB9A P51151 1/20 0.41
GFER P55789 1/20 0.41
COMT P21964 1/20 0.41
NR3C2 P08235 1/20 0.41
HRH3 Q9Y5N1 1/20 0.40
CYP19A1 P11511 1/20 0.39
CYP1A2 P05177 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27752733 0.83 NOS1 (0.40) TAAR1NOS1NOS2ALDH1A1SMN1; SMN2
SCHEMBL3947954 0.83 TAAR1 (0.51) TAAR1DAONOS1MPOIDO1
SCHEMBL3947733 0.82 COMT (0.49) TAAR1DAOGPR84NPC1MAPT
SCHEMBL4012117 0.81 TAAR1 (0.50) TAAR1ALDH1A1IDO1
SCHEMBL4012249 0.81 TAAR1 (0.54) TAAR1DAOIDO1
SCHEMBL4012148 0.79 DHFR (0.46) TAAR1DAOALDH1A1NPC1MAPT
SCHEMBL4009916 0.78 NOS1 (0.42) NOS1NOS2SMN1; SMN2NPC1MAPT
SCHEMBL3939288 0.78 MPO (0.46) NOS1NOS2ALDH1A1MPOIDO1
SCHEMBL3932643 0.76 KDR (0.42) SMN1; SMN2NPC1MAPTRAB9AGFER
SCHEMBL3940447 0.76 DRD2 (0.39)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2044063-A1 PYRIMIDINE DERIVATIVES USEFUL IN THE TREATMENT OF CANCER Astra Zeneca AB (SE) 2009-04-08 EP disclosed
WO-2008001070-A1 PYRIMIDINE DERIVATIVES USEFUL IN THE TREATMENT OF CANCER ASTRAZENECA AB (SE) 2008-01-03 WO disclosed
US-20080004302-A1 Novel Compounds ASTRAZENECA AB (SE) 2008-01-03 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080004302-A1 Novel Compounds CYP11B2, CYP11B1, CYP46A1 TAAR1 3903/4885DAO 4285/4885GPR84 794/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.