SCHEMBL4014164

SCHEMBL4014164

c1cnc2c(c1)CCCS2

nearest known ligand 0.40

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SHMT2 P34897 1/20 0.40
TSHR P16473 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.31
CA12 O43570 1/20 0.30
CA1 P00915 1/20 0.30
CA2 P00918 1/20 0.30
CA9 Q16790 1/20 0.30
HTR1A P08908 1/20 0.30
ADRA2A P08913 1/20 0.30
SLC6A2 P23975 1/20 0.30
SLC6A4 P31645 1/20 0.30
KDR P35968 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5475421 1.00 SHMT2 (0.40) SHMT2TSHRL3MBTL1CA12CA1
SCHEMBL674245 0.88
SCHEMBL17892734 0.72 RYR2 (0.53) SHMT2
SCHEMBL6225796 0.68 MAPT (0.47) TSHRHTR1AADRA2ASLC6A2SLC6A4
SCHEMBL31001735 0.68 ALDH1A1 (0.36) SHMT2TSHR
SCHEMBL1399871 0.68
SCHEMBL15539282 0.68 ALDH1A1 (0.36) SHMT2TSHR
SCHEMBL2511410 0.68 HPGD (0.40)
SCHEMBL170259 0.68 SIGMAR1 (0.33)
SCHEMBL26871373 0.67 HRH1 (0.36) SHMT2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2074098-A2 QUINOLINE COMPOUNDS Wyeth (US) 2009-07-01 EP claimed
WO-2008049047-A2 QUINOLINE COMPOUNDS WYETH (US) 2008-04-24 WO claimed