SCHEMBL4014816

SCHEMBL4014816

COC(=O)Oc1c(OC(C)C)nc(-c2ccc(Cl)cc2)nc1C1CC1

nearest known ligand 0.45

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ATM Q13315 1/20 0.45
CNR1 P21554 1/20 0.40
SLC6A3 Q01959 1/20 0.39
PDE4B Q07343 3/20 0.38
PDE4D Q08499 3/20 0.38
ADORA3 P0DMS8 1/20 0.36
IDO1 P14902 5/20 0.35
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
NPC1 O15118 1/20 0.34
LMNA P02545 1/20 0.34
RAB9A P51151 1/20 0.34
NPSR1 Q6W5P4 3/20 0.34
KDM4E B2RXH2 1/20 0.34
HPGD P15428 1/20 0.34
TSHR P16473 1/20 0.34
NAMPT P43490 1/20 0.34
DHPS P49366 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4008876 0.90 ATM (0.48) ATMCNR1SLC6A3PDE4BPDE4D
SCHEMBL4014601 0.84 DHPS (0.42) CNR1SLC6A3PDE4BPDE4DADORA3
SCHEMBL8022478 0.83 ATM (0.46) ATMCNR1SLC6A3PDE4BPDE4D
SCHEMBL4008874 0.81 ATM (0.50) ATMCNR1SLC6A3PDE4BPDE4D
SCHEMBL4010086 0.79 ATM (0.46) ATMCNR1ADORA3MEN1KMT2A
SCHEMBL4009793 0.77 NR1H4 (0.37) ATMCNR1PDE4BPDE4DNAMPT
SCHEMBL4006533 0.75 PDE4B (0.39) SLC6A3PDE4BPDE4DADORA3RAB9A
SCHEMBL8033148 0.74 SLC6A3 (0.48) SLC6A3PDE4BPDE4DMEN1KMT2A
SCHEMBL4009408 0.73 DHPS (0.39) CNR1PDE4BPDE4DADORA3SMN1; SMN2
SCHEMBL8031484 0.72 SLC6A3 (0.42) CNR1SLC6A3PDE4BPDE4DIDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009080248-A1 SUBSTITUTED 2-PHENYLPYRIMIDINE-5-CARBOXYLIC ACIDS AND THE USE THEREOF BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2009-07-02 WO disclosed