SCHEMBL4017565

SCHEMBL4017565

COc1ccc(Cl)c(-c2ccnc3c(Cl)cccc23)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 1/20 0.47
NR1H3 Q13133 1/20 0.47
SMN1; SMN2 Q16637 2/20 0.46
HTT P42858 1/20 0.46
HSD17B10 Q99714 1/20 0.46
CCNT1 O60563 2/20 0.46
CDK9 P50750 2/20 0.46
NR4A2 P43354 1/20 0.45
ALDH1A1 P00352 3/20 0.45
KDM4E B2RXH2 1/20 0.45
HSP90AA1 P07900 1/20 0.44
HSP90AB1 P08238 1/20 0.44
MAPK14 Q16539 2/20 0.42
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
ALOX15 P16050 1/20 0.41
KDM1A O60341 1/20 0.41
CCR1 P32246 1/20 0.40
CCR5 P51681 1/20 0.40
CCR8 P51685 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4013308 0.89 HTR1A (0.47) NR1H2NR1H3SMN1; SMN2CCNT1CDK9
SCHEMBL4013857 0.86 NR1H2 (0.47) NR1H2NR1H3CCNT1CDK9ALOX15
SCHEMBL4011959 0.85 LRRK2 (0.42) NR1H2NR1H3CCNT1CDK9ALDH1A1
SCHEMBL4011482 0.84 NR1H2 (0.47) NR1H2NR1H3HTTCCNT1CDK9
SCHEMBL2449164 0.80 HSP90AA1 (0.43) SMN1; SMN2HTTHSD17B10ALDH1A1KDM4E
SCHEMBL4013124 0.80 NR4A2 (0.51) SMN1; SMN2HTTNR4A2HSP90AA1HSP90AB1
SCHEMBL4012080 0.79 NR1H2 (0.47) NR1H2NR1H3SMN1; SMN2NR4A2ALDH1A1
SCHEMBL4020515 0.79 NR1H2 (0.78) NR1H2NR1H3
SCHEMBL4011946 0.78 NR4A2 (0.49) NR1H2NR1H3SMN1; SMN2HTTHSD17B10
SCHEMBL4018332 0.77 NR1H2 (0.63) NR1H2NR1H3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2074098-A2 QUINOLINE COMPOUNDS Wyeth (US) 2009-07-01 EP disclosed
WO-2008049047-A2 QUINOLINE COMPOUNDS WYETH (US) 2008-04-24 WO disclosed