SCHEMBL4019201

SCHEMBL4019201

COC(=O)Oc1cnn2c(NC(C)C)c(-c3ncc(Cl)cc3Cl)c(Cl)nc12

nearest known ligand 0.33

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CRHR1 P34998 3/20 0.33
TYK2 P29597 1/20 0.31
IRAK4 Q9NWZ3 1/20 0.31
CDK2 P24941 1/20 0.31
PDE4B Q07343 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3260212 0.92 CRHR1 (0.33) CRHR1TYK2IRAK4CDK2PDE4B
SCHEMBL3258832 0.87 CRHR1 (0.35) CRHR1TYK2
SCHEMBL2794165 0.85 ALDH1A1 (0.39) CRHR1TYK2IRAK4PDE4B
SCHEMBL2796083 0.84 KDM4E (0.38) TYK2IRAK4PDE4B
SCHEMBL2794767 0.80 IRAK4 (0.37) TYK2IRAK4
SCHEMBL4017079 0.80 CRHR1 (0.35) CRHR1TYK2
SCHEMBL5290255 0.77 CRHR1 (0.38) CRHR1
SCHEMBL3262058 0.73 CYP2C19 (0.37)
SCHEMBL5291917 0.73 CNR1 (0.37) CRHR1
SCHEMBL5768799 0.70 EGLN2 (0.37) IRAK4CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2014661-A1 Hererocyclically substituted heterocyclic carboxylic acid derivates Bayer CropScience AG (DE) 2009-01-14 EP disclosed