SCHEMBL4017079

SCHEMBL4017079

COC(=O)Oc1cnn2c(O)c(-c3ncc(Cl)cc3Cl)c(O)nc12

nearest known ligand 0.35

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CRHR1 P34998 3/20 0.35
TYK2 P29597 1/20 0.31
MRGPRX4 Q96LA9 1/20 0.31
ALDH1A1 P00352 2/20 0.30
KDM4E B2RXH2 1/20 0.30
USP2 O75604 1/20 0.30
HSD17B10 Q99714 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3258832 0.84 CRHR1 (0.35) CRHR1TYK2MRGPRX4ALDH1A1KDM4E
SCHEMBL5283300 0.83 CRHR1 (0.37) CRHR1MRGPRX4KDM4E
SCHEMBL2796946 0.83 ALDH1A1 (0.42) CRHR1TYK2MRGPRX4ALDH1A1KDM4E
SCHEMBL4019201 0.80 CRHR1 (0.33) CRHR1TYK2
SCHEMBL5324293 0.74 KDM4E (0.43) CRHR1ALDH1A1KDM4EHSD17B10
SCHEMBL3260212 0.72 CRHR1 (0.33) CRHR1TYK2
SCHEMBL5291917 0.69 CNR1 (0.37) CRHR1MRGPRX4
SCHEMBL5771022 0.69 MEN1 (0.33) ALDH1A1
SCHEMBL3265665 0.69 PDE4A (0.31)
SCHEMBL5774361 0.68 CDK4 (0.32) ALDH1A1KDM4EHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2014661-A1 Hererocyclically substituted heterocyclic carboxylic acid derivates Bayer CropScience AG (DE) 2009-01-14 EP disclosed