SCHEMBL3262058

SCHEMBL3262058

COC(=O)Oc1cnn2c(NC(C)C)c(-n3nc(C)cc3C)c(Cl)nc12

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 2/20 0.37
LMNA P02545 2/20 0.37
NPSR1 Q6W5P4 2/20 0.37
CYP1A2 P05177 1/20 0.37
MAPT P10636 1/20 0.36
HPGD P15428 1/20 0.36
ALDH1A1 P00352 3/20 0.34
L3MBTL1 Q9Y468 3/20 0.34
HSD17B10 Q99714 2/20 0.34
KDM4E B2RXH2 2/20 0.34
USP2 O75604 1/20 0.34
ADORA2A P29274 7/20 0.33
ADORA1 P30542 5/20 0.33
CYP3A4 P08684 4/20 0.33
KCNH2 Q12809 1/20 0.33
MEN1 O00255 1/20 0.32
CYP2C9 P11712 1/20 0.32
KMT2A Q03164 1/20 0.32
HTT P42858 1/20 0.32
ALOX15 P16050 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4018674 0.92 NPSR1 (0.37) CYP2C19LMNANPSR1CYP1A2MAPT
SCHEMBL3257816 0.87 KDM4E (0.36) CYP2C19LMNAMAPTHPGDALDH1A1
SCHEMBL2792537 0.85 KDM4E (0.42) CYP2C19LMNANPSR1CYP1A2MAPT
SCHEMBL2795809 0.84 KDM4E (0.48) CYP2C19LMNANPSR1CYP1A2MAPT
SCHEMBL2796620 0.80 ALDH1A1 (0.38) CYP2C19LMNANPSR1CYP1A2MAPT
SCHEMBL4017611 0.78 KDM4E (0.35) CYP2C19LMNANPSR1CYP1A2MAPT
SCHEMBL4019201 0.73 CRHR1 (0.33)
SCHEMBL2795766 0.70 KDM4E (0.46) CYP2C19LMNACYP1A2MAPTHPGD
SCHEMBL3258768 0.69 LMNA (0.35) LMNAMAPTHPGDALDH1A1L3MBTL1
SCHEMBL5776597 0.68 HTR2C (0.32)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2158204-A2 HETEROCYCLICALLY SUBSTITUTED HETEROCYCLYL CARBOXYLIC ACID DERIVATIVES Bayer CropScience AG (DE) 2010-03-03 EP disclosed
EP-2014661-A1 Hererocyclically substituted heterocyclic carboxylic acid derivates Bayer CropScience AG (DE) 2009-01-14 EP disclosed
WO-2008151735-A2 HETEROCYCLICALLY SUBSTITUTED HETEROCYCLYL CARBOXYLIC ACID DERIVATIVES BAYER CROPSCIENCE AG (DE) 2008-12-18 WO disclosed