SCHEMBL4024265

SCHEMBL4024265

NC(=O)c1ccc(Oc2ccc(C(N)C3Cc4ccccc4C3)cc2F)cc1O

nearest known ligand 0.38

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PNLIP P16233 1/20 0.38
PARP10 Q53GL7 5/20 0.36
PARP15 Q460N3 2/20 0.34
PARP14 Q460N5 1/20 0.34
PARG Q86W56 1/20 0.34
LMNA P02545 1/20 0.33
HTT P42858 1/20 0.33
OPRK1 P41145 6/20 0.33
OPRM1 P35372 5/20 0.33
OPRD1 P41143 5/20 0.33
UGCG Q16739 1/20 0.32
CTNNB1 P35222 1/20 0.32
SCN3A Q9NY46 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4020001 0.88 PARP10 (0.33) PARP10PARP15PARP14LMNASCN3A
SCHEMBL4024269 0.77 LMNA (0.42) PNLIPLMNAHTTOPRK1OPRM1
SCHEMBL4020004 0.69 FYN (0.42) PARP10PARP15PARP14LMNAHTT
SCHEMBL4019651 0.67 PARP10 (0.40) PARP10PARP15LMNAHTTOPRK1
SCHEMBL2988681 0.67 PARP10 (0.37) PARP10LMNAOPRK1OPRM1OPRD1
SCHEMBL2707659 0.66 CTNNB1 (0.59) LMNAHTTCTNNB1
SCHEMBL4017274 0.65 PPARD (0.39) PARP10PARP15LMNAHTTOPRK1
SCHEMBL4024256 0.65 DRD4 (0.46) LMNAHTTOPRK1OPRM1OPRD1
SCHEMBL4017097 0.65 PPARD (0.42) LMNAHTT
SCHEMBL4014189 0.64 ROCK2 (0.40) PARP10PARP15LMNAHTTOPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7618996-B2 Diaryl ether derivatives and uses thereof PFIZER INC. (US) 2009-11-17 US claimed
EP-2064199-A1 DIARYL ETHER DERIVATIVES AND USES THEREOF Pfizer Products Inc. (US) 2009-06-03 EP claimed
US-20080070887-A1 Diaryl Ether Derivatives and Uses Thereof PFIZER INC 2008-03-20 US claimed
WO-2008032156-A1 DIARYL ETHER DERIVATIVES AND USES THEREOF PFIZER PRODUCTS INC. (US) 2008-03-20 WO claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080070887-A1 Diaryl Ether Derivatives and Uses Thereof OPRD1, OPRK1, OPRL1 PNLIP 1763/4885PARP10 2285/4885PARP15 3250/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.